2. GPCR/G Protein
  3. Endothelin Receptor
  4. BQ-3020 ammonium

BQ-3020 ammonium is a selective endothelin receptor (ETB receptor) agonist. BQ-3020 ammonium inhibits [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 ammonium elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 ammonium makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research. .

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BQ-3020 ammonium Chemical Structure

BQ-3020 ammonium Chemical Structure

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Based on 1 publication(s) in Google Scholar

Other Forms of BQ-3020 ammonium:

BQ-3020 ammonium Related Antibodies

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Description

BQ-3020 ammonium is a selective endothelin receptor (ETB receptor) agonist. BQ-3020 ammonium inhibits [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 ammonium elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 ammonium makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research[1][2]. .

Molecular Weight

2006.32 (free base)

Formula

C96H140N20O25S.xNH3
Appearance

Solid

Color

White to off-white

Sequence

Ac-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp
Sequence Shortening

Ac-LMDKEAVYFAHLDIIW
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Sealed storage, away from moisture and light, under nitrogen

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light, under nitrogen)

Solvent & Solubility
In Vitro: 

DMSO : 5 mg/mL (Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

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This equation is commonly abbreviated as: C1V1 = C2V2

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Purity & Documentation
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BQ-3020 ammonium Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

BQ-3020BQ3020BQ 3020Endothelin ReceptorETB receptor agonistvasoconstrictioncardiovascular diseaseendothelin receptorcancer painInhibitorinhibitorinhibit

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BQ-3020 ammonium
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