2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. CB2 modulator 1

CB2 modulator 1 (compound 130) is a potent CB2 modulator. CB2 modulator 1 has the potential for immunedisorders, inflammation, osteoporosis, renal ischemia.

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CB2 modulator 1 Chemical Structure

CB2 modulator 1 Chemical Structure

CAS No. : 666261-80-9

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Based on 1 publication(s) in Google Scholar

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Description

CB2 modulator 1 (compound 130) is a potent CB2 modulator. CB2 modulator 1 has the potential for immunedisorders, inflammation, osteoporosis, renal ischemia[1].

IC50 & Target[1]

CB2

 

Molecular Weight

380.36

Formula

C18H19F3N4O2
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(C1=CN=C(NC2=CC=CC=C2)N=C1C(F)(F)F)NCC3CCOCC3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (262.91 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6291 mL 13.1454 mL 26.2909 mL
5 mM 0.5258 mL 2.6291 mL 5.2582 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

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(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Purity: 99.75%

SDS (251 KB)

COA (246 KB) HNMR (136 KB) LCMS (105 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.6291 mL 13.1454 mL 26.2909 mL 65.7272 mL
5 mM 0.5258 mL 2.6291 mL 5.2582 mL 13.1454 mL
10 mM 0.2629 mL 1.3145 mL 2.6291 mL 6.5727 mL
15 mM 0.1753 mL 0.8764 mL 1.7527 mL 4.3818 mL
20 mM 0.1315 mL 0.6573 mL 1.3145 mL 3.2864 mL
25 mM 0.1052 mL 0.5258 mL 1.0516 mL 2.6291 mL
30 mM 0.0876 mL 0.4382 mL 0.8764 mL 2.1909 mL
40 mM 0.0657 mL 0.3286 mL 0.6573 mL 1.6432 mL
50 mM 0.0526 mL 0.2629 mL 0.5258 mL 1.3145 mL
60 mM 0.0438 mL 0.2191 mL 0.4382 mL 1.0955 mL
80 mM 0.0329 mL 0.1643 mL 0.3286 mL 0.8216 mL
100 mM 0.0263 mL 0.1315 mL 0.2629 mL 0.6573 mL
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CB2 modulator 1 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CB2 modulator 1666261-80-9Cannabinoid ReceptorCB2immunedisordersinflammationosteoporosisrenalischemiaInhibitorinhibitorinhibit

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