2. GPCR/G Protein Neuronal Signaling
  3. Dopamine Receptor
  4. Fluoroclebopride

Fluoroclebopride binds reversibly to dopamine receptors. 18F labeled fluoroclebopride has been used as a probe for studying D2/D3 receptor availability via PET in various monkey models.

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Fluoroclebopride Chemical Structure

Fluoroclebopride Chemical Structure

CAS No. : 154540-49-5

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Based on 1 publication(s) in Google Scholar

Fluoroclebopride Related Antibodies

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Description

Fluoroclebopride binds reversibly to dopamine receptors. 18F labeled fluoroclebopride has been used as a probe for studying D2/D3 receptor availability via PET in various monkey models[1][2].

Molecular Weight

391.87

Formula

C20H23ClFN3O2
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(NC1CCN(CC2=CC=C(F)C=C2)CC1)C3=CC(Cl)=C(N)C=C3OC
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : ≥ 125 mg/mL (318.98 mM; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.5519 mL 12.7593 mL 25.5187 mL
5 mM 0.5104 mL 2.5519 mL 5.1037 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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Volume (start)

V1

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C2

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V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.5519 mL 12.7593 mL 25.5187 mL 63.7967 mL
5 mM 0.5104 mL 2.5519 mL 5.1037 mL 12.7593 mL
10 mM 0.2552 mL 1.2759 mL 2.5519 mL 6.3797 mL
15 mM 0.1701 mL 0.8506 mL 1.7012 mL 4.2531 mL
20 mM 0.1276 mL 0.6380 mL 1.2759 mL 3.1898 mL
25 mM 0.1021 mL 0.5104 mL 1.0207 mL 2.5519 mL
30 mM 0.0851 mL 0.4253 mL 0.8506 mL 2.1266 mL
40 mM 0.0638 mL 0.3190 mL 0.6380 mL 1.5949 mL
50 mM 0.0510 mL 0.2552 mL 0.5104 mL 1.2759 mL
60 mM 0.0425 mL 0.2127 mL 0.4253 mL 1.0633 mL
80 mM 0.0319 mL 0.1595 mL 0.3190 mL 0.7975 mL
100 mM 0.0255 mL 0.1276 mL 0.2552 mL 0.6380 mL
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Fluoroclebopride Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Fluoroclebopride154540-49-5Dopamine ReceptorInhibitorinhibitorinhibit

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