2. GPCR/G Protein
  3. Bradykinin Receptor
  4. Fulimetibant

Fulimetibant is a bradykinin receptor antagonist.

For research use only. We do not sell to patients.

Fulimetibant Chemical Structure

Fulimetibant Chemical Structure

CAS No. : 2231142-90-6

Size Price Stock Quantity
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO
ready for reconstitution
 USD 440 In-stock
Solution
10 mM * 1 mL in DMSO USD 440 In-stock
Solid
5 mg USD 410 In-stock
10 mg USD 670 In-stock
25 mg USD 1350 In-stock
50 mg USD 2200 In-stock
100 mg USD 3580 In-stock
200 mg   Get quote  
500 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

Fulimetibant Related Antibodies

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Bradykinin B1 Receptor (B1R) Bradykinin B2 Receptor (B2R)

  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

Fulimetibant is a bradykinin receptor antagonist[1].

IC50 & Target

Bradykinin receptor[1]
Molecular Weight

487.45

Formula

C25H21F4N3O3
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(C1=C(C2=CN(C3CCC3)N=C2)C=CC(NC(C4(CC4)C5=CC=C(C(F)(F)F)C=C5F)=O)=C1)O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (205.15 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.0515 mL 10.2575 mL 20.5149 mL
5 mM 0.4103 mL 2.0515 mL 4.1030 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.0515 mL 10.2575 mL 20.5149 mL 51.2873 mL
5 mM 0.4103 mL 2.0515 mL 4.1030 mL 10.2575 mL
10 mM 0.2051 mL 1.0257 mL 2.0515 mL 5.1287 mL
15 mM 0.1368 mL 0.6838 mL 1.3677 mL 3.4192 mL
20 mM 0.1026 mL 0.5129 mL 1.0257 mL 2.5644 mL
25 mM 0.0821 mL 0.4103 mL 0.8206 mL 2.0515 mL
30 mM 0.0684 mL 0.3419 mL 0.6838 mL 1.7096 mL
40 mM 0.0513 mL 0.2564 mL 0.5129 mL 1.2822 mL
50 mM 0.0410 mL 0.2051 mL 0.4103 mL 1.0257 mL
60 mM 0.0342 mL 0.1710 mL 0.3419 mL 0.8548 mL
80 mM 0.0256 mL 0.1282 mL 0.2564 mL 0.6411 mL
100 mM 0.0205 mL 0.1026 mL 0.2051 mL 0.5129 mL
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Fulimetibant Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Fulimetibant2231142-90-6Bradykinin ReceptorInhibitorinhibitorinhibit

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