1. Cell Cycle/DNA Damage Metabolic Enzyme/Protease Epigenetics
  2. HSP Histone Demethylase
  3. HSP90/LSD1-IN-1

HSP90/LSD1-IN-1 (compound 6) is a HSP90/LSD1 dual inhibitor. HSP90/LSD1-IN-1 inhibits the proliferation of prostate cancer cell lines PC-3 and DU145, with GI50 values ​​of 0.24 and 0.30 μM, respectively.

For research use only. We do not sell to patients.

HSP90/LSD1-IN-1 Chemical Structure

HSP90/LSD1-IN-1 Chemical Structure

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Description

HSP90/LSD1-IN-1 (compound 6) is a HSP90/LSD1 dual inhibitor. HSP90/LSD1-IN-1 inhibits the proliferation of prostate cancer cell lines PC-3 and DU145, with GI50 values ​​of 0.24 and 0.30 μM, respectively[1].

IC50 & Target

HSP90

 

LSD1

 

Molecular Weight

380.48

Formula

C23H28N2O3

SMILES

O=C(N(CC)C1=CC=CC(CN(C)CC#C)=C1)C2=CC(C(C)C)=C(O)C=C2O

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
HSP90/LSD1-IN-1
Cat. No.:
HY-169098
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