1. Signaling Pathways
  2. Epigenetics
  3. Histone Demethylase
  4. Histone Demethylase Inhibitors

Histone Demethylase Inhibitors

KDM1/LSD1

KDM2

KDM3

KDM4

KDM5

KDM6

KDM7

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Histone Demethylase Inhibitors & Antagonists
Product Name KDM1/LSD1 KDM2 KDM3 KDM4 KDM5 KDM6 KDM7 Purity
GSK-J4          
KDM6
  99.64%
IOX1  
KDM2
KDM3
KDM4
 
KDM6
  99.72%
GSK2879552
KDM1/LSD1
            99.75%
LSD1/HDAC6-IN-2
LSD1, IC50: 5 nM
            99.66%
LSD1-IN-31
LSD1
           
LSD1-IN-34
LSD1, IC50: 4.51 nM
           
CPI-455        
KDM5
    98.95%
JIB-04      
KDM4
KDM5
KDM6
  98.29%
GSK-J1          
KDM6
  99.94%
QC6352      
KDM4A, IC50: 104 nM
KDM4B, IC50: 56 nM
KDM4C, IC50: 35 nM
KDM4D, IC50: 104 nM
KDM5B, IC50: 750 nM
    99.48%
KDM5-C70        
KDM5
   
Tranylcypromine hemisulfate
KDM1/LSD1
            99.94%
SP2509
KDM1/LSD1
            99.90%
Seclidemstat
KDM1/LSD1
            99.77%
GSK-J4 hydrochloride          
KDM6
  98.83%
GSK467        
KDM5, Ki: 10 nM
KDM5, IC50: 26 nM
    99.55%
Pulrodemstat benzenesulfonate
KDM1/LSD1
            99.12%
NCGC00244536      
KDM4
      99.58%
AS8351        
KDM5
    99.19%
KDOAM-25 citrate        
KDM5
    98.11%
Daminozide  
KDM2
          99.79%
Bomedemstat hydrochloride
KDM1/LSD1
            99.94%
KDM5A-IN-1        
KDM5
    99.80%
ML324      
KDM4
      98.54%
PFI-90    
KDM3
        99.86%
KDM2A/7A-IN-1  
KDM2
          99.94%
KDM5-IN-1        
KDM5
    99.87%
Bomedemstat dihydrochloride
KDM1/LSD1
            99.55%
TK-129        
KDM5, IC50: 44 nM
    ≥98.0%
PBIT        
KDM5
    99.46%
GSK 690 Hydrochloride
KDM1/LSD1
            98.58%
S2101
KDM1/LSD1
            99.73%
KDM2/7-IN-1  
KDM2
 
KDM4
   
KDM7
99.00%
YUKA1        
KDM5
    99.56%
KDM4C-IN-1      
KDM4
      98.99%
INCB059872 dihydrochloride
KDM1/LSD1
            99.18%
KDM2B-IN-4  
KDM2
          99.59%
Iadademstat
LSD1
            99.61%
JQKD82 trihydrochloride        
KDM5
    99.94%
DDP-38003 dihydrochloride
KDM1/LSD1
            98.22%
HDAC6-IN-3
KDM1/LSD1
            ≥98.0%
LSD1-IN-30
LSD1, IC50: 0.291 μM
            99.03%
CBB1007 trihydrochloride
KDM1/LSD1
           
Pulrodemstat
KDM1/LSD1
           
Bomedemstat
KDM1/LSD1
            99.55%
INCB059872
KDM1/LSD1
            98.06%
KDM4-IN-2      
KDM4
      98.29%
CBB1007 hydrochloride
KDM1/LSD1
            ≥98.0%
LSD1-IN-5
KDM1/LSD1
           
LSD1-IN-6
KDM1/LSD1
           
Pulrodemstat Methylbenzenesulfonate
KDM1/LSD1
           
CPI-455 hydrochloride        
KDM5
   
LSD1/HDAC6-IN-1
KDM1/LSD1
           
LSD1-IN-13 hydrochloride
KDM1/LSD1
           
MC2652
KDM1/LSD1
           
KDM4-IN-4      
KDM4A-Tudor domain, Ki: 80 μM
     
HSP90/LSD1-IN-1
LSD1
           
LSD1-UM-109
LSD1, IC50: 3.1 nM
           
S1427
KDM1/LSD1
           
LSD1-IN-23
KDM1/LSD1, IC50: 0.58 μM
           
LSD1/2-IN-4
KDM1/LSD1
           
NCL1
LSD1, IC50: 2.5 ± 0.5 μM
           
cis-4-Br-2,5-F2-PCPA
KDM1/LSD1
           
KDM1/CDK1-IN-1
KDM1/LSD1
           
LSD1-IN-26
LSD1, IC50: 25.3 ± 1.4 nM
           
LSD1-IN-21
LSD1, IC50: 0.956 μM
           
KDM5-C49        
KDM5
   
LSD1-IN-35
LSD1
           
LSD1-IN-18
KDM1/LSD1
           
LSD1-IN-25
LSD1, IC50: 46 nM
LSD1, Ki: 30.3 nM
           
(1S,2R)-Tranylcypromine hydrochloride
KDM1/LSD1
           
Arborinine
LSD1
           
LSD1-IN-22
KDM1/LSD1
           
LSD1-IN-19
KDM1/LSD1
           
LSD1/2-IN-3
KDM1/LSD1
           
Tranylcypromine-d5 hydrochloride
KDM1/LSD1
           
LSD1/HDAC-IN-1
LSD1, IC50: 0.571 μM
           
JQKD82        
KDM5
   
LSD1/ER-IN-1
KDM1/LSD1
           
LSD1-IN-36
LSD1, IC50: 0.8 nM
           
CBB1003 hydrochloride
KDM1/LSD1
           
GSK-J1 lithium salt          
KDM6
  98.26%