2. Metabolic Enzyme/Protease
  3. Glutaminase
  4. hTG2 inhibitor VA4

hTG2 inhibitor VA4 (compound VA4) is an irreversible Type 2 transglutaminase (TG2) inhibitor. hTG2 inhibitor VA4 reacts exclusively at the TG2 transamidase site, inhibits both transamidase and GTP-binding activities.

For research use only. We do not sell to patients.

hTG2 inhibitor VA4 Chemical Structure

hTG2 inhibitor VA4 Chemical Structure

CAS No. : 2088001-23-2

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hTG2 inhibitor VA4 Related Antibodies

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Description

hTG2 inhibitor VA4 (compound VA4) is an irreversible Type 2 transglutaminase (TG2) inhibitor. hTG2 inhibitor VA4 reacts exclusively at the TG2 transamidase site, inhibits both transamidase and GTP-binding activities[1].

In Vitro

hTG2 inhibitor VA4 (compound VA4) suppress ECS cell (Epidermal cancer stem cells) spheroid formation and invasion[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

hTG2 inhibitor VA4 Related Antibodies
Molecular Weight

635.77

Formula

C33H41N5O6S
CAS No.
SMILES

O=C(OCC1=CC=CC=C1)N[C@H](C(N2CCN(S(=O)(C3=C4C=CC=C(N(C)C)C4=CC=C3)=O)CC2)=O)CCCCNC(C=C)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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hTG2 inhibitor VA4 Related Classifications

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  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

hTG2 inhibitor VA42088001-23-2GlutaminaseTransglutaminaseECS cellInhibitorinhibitorinhibit

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hTG2 inhibitor VA4
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HY-122709
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