1. GPCR/G Protein Neuronal Signaling
  2. 5-HT Receptor Adrenergic Receptor Dopamine Receptor
  3. Iloperidone carboxylic acid

Iloperidone carboxylic acid  (Synonyms: P95-12113)

Cat. No.: HY-W741575
Data Sheet Handling Instructions Technical Support

Iloperidone carboxylic acid (P95-12113) is the metabolite of Iloperidone (HY-17410). Iloperidone carboxylic acid exhibits good affinity for 5-HT2A receptor with pKi of 8.15, and moderate affinity for adrenergic receptor α1/α2B/α2C.

For research use only. We do not sell to patients.

Iloperidone carboxylic acid Chemical Structure

Iloperidone carboxylic acid Chemical Structure

CAS No. : 475110-48-6

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Description

Iloperidone carboxylic acid (P95-12113) is the metabolite of Iloperidone (HY-17410). Iloperidone carboxylic acid exhibits good affinity for 5-HT2A receptor with pKi of 8.15, and moderate affinity for adrenergic receptor α1/α2B/α2C[1].

IC50 & Target

Human 5-HT2A Receptor

8.15 (pKi)

rat α1-adrenergic receptor

7.67 (pKi)

human α2C-adrenoceptor

7.32 (pKi)

human α2B-adrenoceptor

7.08 (pKi)

human α2A-adrenoceptor

6.42 (pKi)

Rat D3 Receptor

6.11 (pKi)

Human D1 Receptor

5.94 (pKi)

Human 5-HT6 Receptor

5.59 (pKi)

Molecular Weight

428.45

Formula

C23H25FN2O5

CAS No.
SMILES

COC1=C(OCCCN2CCC(C3=NOC4=C3C=CC(F)=C4)CC2)C=CC(C(O)=O)=C1

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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Iloperidone carboxylic acid
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HY-W741575
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