2. Metabolic Enzyme/Protease GPCR/G Protein Anti-infection Neuronal Signaling Autophagy Membrane Transporter/Ion Channel Immunology/Inflammation
  3. Dopamine Receptor Enterovirus 5-HT Receptor Autophagy Calcium Channel Histamine Receptor Cytochrome P450
  4. Levomepromazine maleate

Levomepromazine maleate  (Synonyms: Methotrimeprazine maleate)

Cat. No.: HY-W344044 Purity: 99.92%
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Levomepromazine maleate (Methotrimeprazine maleate) is an N-substituted phenylthiazine antipsychotic sedative that blocks multiple receptors. Levomepromazine maleate is a potent inhibitor of CYP2D6 and is useful in the study of schizophreni.

For research use only. We do not sell to patients.

Levomepromazine maleate Chemical Structure

Levomepromazine maleate Chemical Structure

CAS No. : 7104-38-3

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Other Forms of Levomepromazine maleate:

Levomepromazine maleate Related Antibodies

Top Publications Citing Use of Products

1 Publications Citing Use of MCE Levomepromazine maleate

View All Dopamine Receptor Isoform Specific Products:

View All Isoforms
Dopamine Receptor D1 Receptor D2 Receptor D3 Receptor D4 Receptor D5 Receptor

View All Calcium Channel Isoform Specific Products:

View All Isoforms
N-type calcium channel L-type calcium channel P/Q-type calcium channel T-type calcium channel Calcium Channel

View All Histamine Receptor Isoform Specific Products:

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H1 Receptor H2 Receptor H3 Receptor H4 Receptor Histamine Receptor

View All Cytochrome P450 Isoform Specific Products:

View All Isoforms
CYP1 CYP2 CYP3 CYP4 CYP11 CYP17 Aromatase/CYP19A1 CYP26 CYP51 CYP1A2 CYP2D6 CYP2C9 CYP2C19 CYP3A4 CYP17A1

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Description

Levomepromazine maleate (Methotrimeprazine maleate) is an N-substituted phenylthiazine antipsychotic sedative that blocks multiple receptors. Levomepromazine maleate is a potent inhibitor of CYP2D6 and is useful in the study of schizophreni[1][2].

Molecular Weight

444.54

Formula

C23H28N2O5S
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

CN(C)C[C@@H](C)CN1C2=CC(OC)=CC=C2SC3=CC=CC=C31.OC(/C=C\C(O)=O)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 50 mg/mL (112.48 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2495 mL 11.2476 mL 22.4952 mL
5 mM 0.4499 mL 2.2495 mL 4.4990 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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C2

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V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.2495 mL 11.2476 mL 22.4952 mL 56.2379 mL
5 mM 0.4499 mL 2.2495 mL 4.4990 mL 11.2476 mL
10 mM 0.2250 mL 1.1248 mL 2.2495 mL 5.6238 mL
15 mM 0.1500 mL 0.7498 mL 1.4997 mL 3.7492 mL
20 mM 0.1125 mL 0.5624 mL 1.1248 mL 2.8119 mL
25 mM 0.0900 mL 0.4499 mL 0.8998 mL 2.2495 mL
30 mM 0.0750 mL 0.3749 mL 0.7498 mL 1.8746 mL
40 mM 0.0562 mL 0.2812 mL 0.5624 mL 1.4059 mL
50 mM 0.0450 mL 0.2250 mL 0.4499 mL 1.1248 mL
60 mM 0.0375 mL 0.1875 mL 0.3749 mL 0.9373 mL
80 mM 0.0281 mL 0.1406 mL 0.2812 mL 0.7030 mL
100 mM 0.0225 mL 0.1125 mL 0.2250 mL 0.5624 mL
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Levomepromazine maleate Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Levomepromazine7104-38-3MethotrimeprazineDopamine ReceptorEnterovirus5-HT ReceptorAutophagyCalcium ChannelHistamine ReceptorCytochrome P450RhinovirusHRVHRVsHEVHEVsSerotonin Receptor5-hydroxytryptamine ReceptorCa2+ channelsCa channelsCYPsCalmantipsychoticreceptor blockingschizophreniaInhibitorinhibitorinhibit

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