1. Metabolic Enzyme/Protease
  2. Carboxypeptidase
  3. Mergetpa

Mergetpa is a carboxypeptidase inhibitor used to block the conversion of kinins and B2 receptor antagonists to metabolites lacking the C-terminal arginine.

For research use only. We do not sell to patients.

Mergetpa Chemical Structure

Mergetpa Chemical Structure

CAS No. : 77102-28-4

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5 mg USD 278 In-stock
10 mg USD 445 In-stock
25 mg USD 895 In-stock
50 mg USD 1438 In-stock
100 mg USD 2300 In-stock
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Based on 1 publication(s) in Google Scholar

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Description

Mergetpa is a carboxypeptidase inhibitor used to block the conversion of kinins and B2 receptor antagonists to metabolites lacking the C-terminal arginine[1].

Molecular Weight

237.34

Formula

C7H15N3O2S2

CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O=C(C(CSCCNC(N)=N)CS)O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, stored under nitrogen, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen, away from moisture)

Solvent & Solubility
In Vitro: 

H2O : 15 mg/mL (63.20 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 4.2134 mL 21.0668 mL 42.1336 mL
5 mM 0.8427 mL 4.2134 mL 8.4267 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (stored under nitrogen, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

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Volume (start)

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Concentration (final)

C2

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Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
The concentration of the stock solution you require exceeds the measured solubility. The following solution is for reference only.If necessary, please contact MedChemExpress (MCE).
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (stored under nitrogen, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
H2O 1 mM 4.2134 mL 21.0668 mL 42.1336 mL 105.3341 mL
5 mM 0.8427 mL 4.2134 mL 8.4267 mL 21.0668 mL
10 mM 0.4213 mL 2.1067 mL 4.2134 mL 10.5334 mL
15 mM 0.2809 mL 1.4045 mL 2.8089 mL 7.0223 mL
20 mM 0.2107 mL 1.0533 mL 2.1067 mL 5.2667 mL
25 mM 0.1685 mL 0.8427 mL 1.6853 mL 4.2134 mL
30 mM 0.1404 mL 0.7022 mL 1.4045 mL 3.5111 mL
40 mM 0.1053 mL 0.5267 mL 1.0533 mL 2.6334 mL
50 mM 0.0843 mL 0.4213 mL 0.8427 mL 2.1067 mL
60 mM 0.0702 mL 0.3511 mL 0.7022 mL 1.7556 mL

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

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Mergetpa Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Mergetpa
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HY-W704574
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