2. Epigenetics
  3. Epigenetic Reader Domain
  4. pan-BET/BD2-IN-1

pan-BET/BD2-IN-1 (compound 6b) is a selective extra-terminal (BET) protein inhibitor (BRDT-1 Ki = 1.05 μM and BRD4-1 Ki = 0.68 μM). pan-BET/BD2-IN-1 inhibits MM.1S cancer cell growth with an IC50 of 2.6 μM.

For research use only. We do not sell to patients.

pan-BET/BD2-IN-1 Chemical Structure

pan-BET/BD2-IN-1 Chemical Structure

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Description

pan-BET/BD2-IN-1 (compound 6b) is a selective extra-terminal (BET) protein inhibitor (BRDT-1 Ki = 1.05 μM and BRD4-1 Ki = 0.68 μM). pan-BET/BD2-IN-1 inhibits MM.1S cancer cell growth with an IC50 of 2.6 μM[1].

Molecular Weight

489.52

Formula

C27H27N3O6
SMILES

CC1=CC=C(C(OCCOC2=C(C=CC=C2)COC3=O)=C1)C4C3=C(NC(N(C(N5)=O)CC)=C4C5=O)C
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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pan-BET/BD2-IN-1 Related Classifications

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Keywords:

pan-BET/BD2-IN-1Epigenetic Reader Domainextra-terminal (BET) proteinMM.1SBRD4-1BRDT-1Inhibitorinhibitorinhibit

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