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PCAF-IN-1 is a highly selective PCAF inhibitor. PCAF-IN-1 is a antitumor agents, which can be used in tumor research research.

For research use only. We do not sell to patients.

PCAF-IN-1 Chemical Structure

PCAF-IN-1 Chemical Structure

CAS No. : 2439194-86-0

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Based on 1 publication(s) in Google Scholar

PCAF-IN-1 Related Antibodies

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Description

PCAF-IN-1 is a highly selective PCAF inhibitor. PCAF-IN-1 is a antitumor agents, which can be used in tumor research research[1].

In Vitro

PCAF-IN-1 (Compound 32) (10 μM, 72 hours; human tumor cell lines) exerts the most potent antitumor activities against human cancer cell lines[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

PCAF-IN-1 Related Antibodies

Cell Cytotoxicity Assay[1]

Cell Line: Hepatocellular carcinoma (HePG-2), breast cancer (MCF-7), prostate cancer (PC3) and colorectal carcinoma (HCT-116).
Concentration: 10 μM
Incubation Time: 72 hours
Result: Inhibited with IC50 values of 4.89, 6.18, 9.71 and 3.76 μM for HePG-2, MCF-7, PC3 and HCT-116, respectively.
Molecular Weight

310.74

Formula

C15H11ClN6
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

NNC1=NN2C(C3=CC=C(C=C3)Cl)=NN=C2C4=CC=CC=C41
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 0.5 mg/mL (1.61 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 3.2181 mL 16.0906 mL 32.1812 mL
5 mM --- --- ---
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 3.2181 mL 16.0906 mL 32.1812 mL 80.4531 mL
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PCAF-IN-1 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PCAF-IN-12439194-86-0OthersPCAFantitumorMitochondrial pathwayInhibitorinhibitorinhibit

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HY-147894
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