2. PI3K/Akt/mTOR
  3. PDK-1
  4. PKD-IN-1 dihydrochloride

PKD-IN-1 dihydrochloride (compound 32), an aminoethylamino-aryl (AEAA) compound, acts as PKD-1 inhibitor. PKD-IN-1 can be used for protein kinase D (PKD)-mediated diseases research.

For research use only. We do not sell to patients.

PKD-IN-1 dihydrochloride Chemical Structure

PKD-IN-1 dihydrochloride Chemical Structure

CAS No. : 2308510-39-4

Size Price Stock Quantity
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO
ready for reconstitution
 USD 110 In-stock
Solution
10 mM * 1 mL in DMSO USD 110 In-stock
Solid
5 mg USD 100 In-stock
10 mg USD 165 In-stock
25 mg USD 290 In-stock
50 mg USD 470 In-stock
100 mg USD 710 In-stock
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of PKD-IN-1 dihydrochloride:

PKD-IN-1 dihydrochloride Related Antibodies

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Description

PKD-IN-1 dihydrochloride (compound 32), an aminoethylamino-aryl (AEAA) compound, acts as PKD-1 inhibitor. PKD-IN-1 can be used for protein kinase D (PKD)-mediated diseases research[1].

Molecular Weight

415.74

Formula

C18H21Cl3N4O
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

OC1=CC=C(Cl)C=C1C2=NC(NC[C@H](N)CC)=C3C=CC=CC3=N2.[H]Cl.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 35.71 mg/mL (85.90 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.4053 mL 12.0267 mL 24.0535 mL
5 mM 0.4811 mL 2.4053 mL 4.8107 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.4053 mL 12.0267 mL 24.0535 mL 60.1337 mL
5 mM 0.4811 mL 2.4053 mL 4.8107 mL 12.0267 mL
10 mM 0.2405 mL 1.2027 mL 2.4053 mL 6.0134 mL
15 mM 0.1604 mL 0.8018 mL 1.6036 mL 4.0089 mL
20 mM 0.1203 mL 0.6013 mL 1.2027 mL 3.0067 mL
25 mM 0.0962 mL 0.4811 mL 0.9621 mL 2.4053 mL
30 mM 0.0802 mL 0.4009 mL 0.8018 mL 2.0045 mL
40 mM 0.0601 mL 0.3007 mL 0.6013 mL 1.5033 mL
50 mM 0.0481 mL 0.2405 mL 0.4811 mL 1.2027 mL
60 mM 0.0401 mL 0.2004 mL 0.4009 mL 1.0022 mL
80 mM 0.0301 mL 0.1503 mL 0.3007 mL 0.7517 mL
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PKD-IN-1 dihydrochloride Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PKD-IN-12308510-39-4PDK-13-Phosphoinositide-dependent protein kinase 1Inhibitorinhibitorinhibit

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