2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. Procaterol hydrochloride hemihydrate

Procaterol hydrochloride hemihydrate  (Synonyms: OPC 2009 hydrochloride hemihydrate)

Cat. No.: HY-129041 Purity: 99.88%
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Procaterol hydrochloride hemihydrate is an orally active β2 adrenoreceptor agonist. Procaterol hydrochloride hemihydrate can be used for the research of asthma.

For research use only. We do not sell to patients.

Procaterol hydrochloride hemihydrate Chemical Structure

Procaterol hydrochloride hemihydrate Chemical Structure

CAS No. : 81262-93-3

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25 mg USD 390 In-stock
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Based on 1 publication(s) in Google Scholar

Other Forms of Procaterol hydrochloride hemihydrate:

Procaterol hydrochloride hemihydrate Related Antibodies

Top Publications Citing Use of Products

1 Publications Citing Use of MCE Procaterol hydrochloride hemihydrate

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  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

Procaterol hydrochloride hemihydrate is an orally active β2 adrenoreceptor agonist. Procaterol hydrochloride hemihydrate can be used for the research of asthma[1][2][3].

In Vitro

Procaterol hydrochloride hemihydrate (0.1 μM, 24-72 h) decreases rhinovirus infection in human tracheal epithelial cells[4].
Procaterol hydrochloride hemihydrate (0-1 μg/mL, 24/48 h) inhibits IL-1β- and TNF-α-mediated eosinophil chemotactic activity in BEAS-2B cell[5].
procaterol hydrochloride hemihydrate (25-200 nM, 20 h) protects 16HBE cells from H2O2-induced oxidative stress[6].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Procaterol hydrochloride hemihydrate Related Antibodies
In Vivo

Procaterol hydrochloride hemihydrate (1, 3 or 10 μg/mL, inhaled administration) inhibits histamine-induced airflow obstruction and microvascular leakage in guinea-pig airways with allergic inflammation[2].
Procaterol hydrochloride hemihydrate (0.1 mg/kg, i.p.) completely abolishes both the Mch-induced cough in conscious guinea pigs[3].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Allergic inflammatory guinea-pig model[2]
Dosage: 1, 3 or 10 μg/mL
Administration: Inhaled administration
Result: Inhibited histamine-induced airflow obstruction and microvascular leakage.
Molecular Weight

335.82

Formula

C16H23ClN2O3.1/2H2O
CAS No.
Appearance

Solid

Color

White to off-white

SMILES

O[C@H]([C@H](NC(C)C)CC)C1=C(C=CC(N2)=O)C2=C(O)C=C1.Cl.[0.5 H2O]
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

H2O : 25 mg/mL (74.44 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.9778 mL 14.8889 mL 29.7779 mL
5 mM 0.5956 mL 2.9778 mL 5.9556 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

  • Molarity Calculator

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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C2

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V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
This product has good water solubility, please refer to the measured solubility data in water/PBS/Saline for details.
The concentration of the stock solution you require exceeds the measured solubility. The following solution is for reference only.If necessary, please contact MedChemExpress (MCE).
Purity & Documentation

Purity: 99.88%

COA (257 KB) HNMR (295 KB) LCMS (268 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
H2O 1 mM 2.9778 mL 14.8889 mL 29.7779 mL 74.4446 mL
5 mM 0.5956 mL 2.9778 mL 5.9556 mL 14.8889 mL
10 mM 0.2978 mL 1.4889 mL 2.9778 mL 7.4445 mL
15 mM 0.1985 mL 0.9926 mL 1.9852 mL 4.9630 mL
20 mM 0.1489 mL 0.7444 mL 1.4889 mL 3.7222 mL
25 mM 0.1191 mL 0.5956 mL 1.1911 mL 2.9778 mL
30 mM 0.0993 mL 0.4963 mL 0.9926 mL 2.4815 mL
40 mM 0.0744 mL 0.3722 mL 0.7444 mL 1.8611 mL
50 mM 0.0596 mL 0.2978 mL 0.5956 mL 1.4889 mL
60 mM 0.0496 mL 0.2481 mL 0.4963 mL 1.2407 mL

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

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Procaterol hydrochloride hemihydrate Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Procaterol hydrochloride hemihydrate81262-93-3OPC 2009 hydrochloride hemihydrateAdrenergic ReceptorBeta ReceptorAsthmarhinovirusinfectionBEAS-2B16HBEoxidative stresscoughInhibitorinhibitorinhibit

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