2. GPCR/G Protein
  3. Protease Activated Receptor (PAR)
  4. Protease-Activated Receptor-1 antagonist 1

Protease-Activated Receptor-1 antagonist 1 

Cat. No.: HY-143313
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Protease-Activated Receptor-1 antagonist 1 (Compound 13) is a protease-activated receptor-1 (PAR-1) antagonist with the IC50 of 3 nM by FLIPR technology. Protease-Activated Receptor-1 antagonist 1 can be used for the research of thrombotic cardiovascular, myocardial infarction, and peripheral arterial disease.

For research use only. We do not sell to patients.

Protease-Activated Receptor-1 antagonist 1 Chemical Structure

Protease-Activated Receptor-1 antagonist 1 Chemical Structure

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Protease-Activated Receptor-1 antagonist 1 Related Antibodies

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PAR1 PAR2 PAR4

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Description

Protease-Activated Receptor-1 antagonist 1 (Compound 13) is a protease-activated receptor-1 (PAR-1) antagonist with the IC50 of 3 nM by FLIPR technology. Protease-Activated Receptor-1 antagonist 1 can be used for the research of thrombotic cardiovascular, myocardial infarction, and peripheral arterial disease[1].

Molecular Weight

438.47

Formula

C25H24F2N2O3
SMILES

[H][C@]12[C@H]([C@@H](C(F)(C[C@]1(C(O[C@@H]2C)=O)O)F)C)/C=C/C3=CC=C(C=N3)C4=CC=CC(C)=C4C#N
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Protease-Activated Receptor-1 antagonist 1 Related Classifications

  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Protease-Activated Receptor-1 antagonist 1Protease Activated Receptor (PAR)Thrombin receptorsprotease-activated receptorPAR-1 antagonistthrombotic cardiovascularmyocardial infarctionperipheral arterial diseaseInhibitorinhibitorinhibit

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