Protease Activated Receptor (PAR) Inhibitors

PAR1

PAR2

PAR4

Protease Activated Receptor (PAR) Inhibitors, Agonists, Antagonists & Activators

Product Name	PAR1	PAR2	PAR4	Purity
TRAP-6	PAR1, IC₅₀: 96 nM			99.84%
Trypsin		PAR2	PAR4
Vorapaxar	PAR1, Ki: 8.1 nM			99.85%
AZ3451		PAR2, IC₅₀: 23 nM		99.84%
PAR4 antagonist 6			hPAR4, IC₅₀: 134 nM mPAR4, IC₅₀: 150 nM
2-Furoyl-LIGRLO-amide		PAR2		99.87%
SCH79797	PAR1, IC₅₀: 70 nM PAR1, Ki: 35 nM			99.74%
BMS-986120	PAR1		PAR4	98.54%
GB-88		PAR2, IC₅₀: 2 μM		99.05%
Protease-Activated Receptor-2, amide		PAR2		98.73%
AZ8838		PAR2		98.87%
GB-110 hydrochloride		PAR2, EC₅₀: .28 μM		99.83%
Vorapaxar sulfate	PAR1, Ki: 8.1 nM			99.81%
I-191		PAR2		99.14%
Parmodulin 2	PAR1, IC₅₀: .26 μM			99.82%
ENMD-1068 hydrochloride		PAR2		98.33%
PZ-128	PAR1			99.47%
AC-55541		PAR2		99.25%
FSLLRY-NH2 TFA		PAR2		99.43%
TFLLR-NH2(TFA)	PAR1, EC₅₀: 1.9 μM			99.78%
FSLLRY-NH2		PAR2		98.52%
SCH79797 dihydrochloride	PAR1			99.91%
PAR-2-IN-1		PAR2		99.79%
Trypsin (MS grade)		PAR2	PAR4
Protease-Activated Receptor-4			PAR4
Atopaxar	PAR1
tcY-NH2 TFA			PAR4	99.72%
VKGILS-NH2		PAR2		99.81%
Protease-Activated Receptor-1, PAR-1 Agonist	PAR1			98.34%
Protease-Activated Receptor-1, PAR-1 Agonist TFA	PAR1			98.54%
BMS-986141			PAR4, IC₅₀: .4 nM	98.86%
I-287		PAR2		99.02%
iso-TRAP-6	PAR1			99.26%
RWJ-56110 dihydrochloride	PAR1, IC₅₀: .4 μM			99.54%
GB83		PAR2		99.80%
FLLRN	PAR1			98.99%
TFLLR-NH2	PAR1, EC₅₀: 1.9 μM
TRAP-6 amide	PAR1			98.12%
GB-110		PAR2, EC₅₀: .28 μM
FR-171113	PAR1, IC₅₀: .29 μM
AY77		PAR2
PAR4 antagonist 5			PAR4
PAR4 antagonist 4			PAR4, IC₅₀: 14.2 nM
PAR4 antagonist 2			PAR4
PAR4 antagonist 1			PAR4, IC₅₀: 1.8 nM
ENMD-1068		PAR2
Atopaxar hydrochloride	PAR1
K-14585		PAR2
AY254		PAR2, EC₅₀: 2 nM
PAR4 antagonist 3			PAR4, IC₅₀: 26.1 nM
RWJ-56110	PAR1, IC₅₀: .4 μM
Protease-Activated Receptor-1 antagonist 2	PAR1, IC₅₀: 7 nM
2-Furoyl-LIGRLO-amide TFA		PAR2
VKGILS-NH2 TFA		PAR2
tcY-NH2			PAR4
ENMD-1068 hydrobromide		PAR2
P4pal10			PAR4
UDM-001651			PAR4
ML354			PAR4, IC₅₀: 140 nM	98.80%
TRAP-6 amide TFA	PAR1
Atopaxar hydrobromide	PAR1, IC₅₀: 5.1 nM

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