Search Result

Search Result

Results for "

ATAD2 inhibitor

" in MedChemExpress (MCE) Product Catalog:

By Targets:	Apoptosis (1) c-Myc (1) Epigenetic Reader Domain (5)
By Research Areas:	Cancer (3) Metabolic Disease (2)

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

AZ13824374	Epigenetic Reader Domain	Cancer
AZ13824374 is a highly potent and selective *ATAD2* bromodomain inhibitor which shows cellular target engagement and antiproliferative activity in a range of breast cancer models. AZ13824374 inhibits ATAD2 with pIC₅₀s of 8.2 and 6.2 in ATAD2 FRET assay and ATAD2 NanoBRET assay, respectively .

GSK8814	Epigenetic Reader Domain	Cancer
GSK8814 is a potent, selective, and ATAD2/2B bromodomain chemical probe and inhibitor, with a binding constant pK_d=8.1 and a pK_i=8.9 in BROMOscan. GSK8814 binds to ATAD2 and BRD4 BD1 with pIC₅₀s of 7.3 and 4.6, respectively. GSK8814 shows 500-fold selectivity for ATAD2 over BRD4 BD1 .

BAY-850 4 Publications Verification	Epigenetic Reader Domain	Metabolic Disease
BAY-850 is a potent and isoform selective ATPase family AAA domain-containing protein 2 *(ATAD2)* inhibitor, with an IC₅₀ of 166 nM.

trans-BAY-850	Epigenetic Reader Domain	Metabolic Disease
trans-BAY-850 is the trans isomer of BAY-850 (HY-119254). BAY-850 is a potent and isoform selective ATPase family AAA domain-containing protein 2 (ATAD2) inhibitor, with an IC₅₀ of 166 nM.

ATAD2-IN-1	Epigenetic Reader Domain Apoptosis c-Myc	Cancer
ATAD2-IN-1 (compound 19f) is a potent *ATAD2* inhibitor (IC₅₀: 0.27 μM) and can induce apoptosis. ATAD2-IN-1 also inhibits c-Myc activation and BT-549 cell migration .

Inquiry Online

Your information is safe with us. * Required Fields.

MCE Japan Authorized Agent ナミキ商事株式会社コスモ・バイオ株式会社
Salutation			Country or Region *
Applicant Name *			Organization Name *
Department *
Email Address *			Product Name *
Cat. No.			Requested quantity *
Phone Number *
Remarks

MedChemExpress Magic Cece

MedChemExpress: Contact Us; About Us; Headquarters; Distributors; Statement on False Report; Careers

Customer Support: Technical Support; Service; Ordering Information; Easy Return; Shipping Rates & Policies; Intellectual Property Promise

Resources: Free Sample; Resources; Molarity Calculator; Dilution Calculator; Terms & Conditions; Reconstitution Calculator; Specific Activity Calculator; DNA/RNA sequence conversion tools

Subscribe to our E-newsletter

Name
Email *

	Sorry, but the email address you supplied was invalid.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.

Copyright © 2013-2025 MedChemExpress. All Rights Reserved.: Site Map Privacy Policy

Join with us