2. GPCR/G Protein
  3. Oxytocin Receptor
  4. SSR126768A free base

SSR126768A free base is an orally active antagonist for oxytocin receptor, with Ki of 0.44 nM. SSR126768A free base is a tocolytic agent, that antagonizes the Oxytocin (HY-17571)-induced intracellular Ca2+ increase and prostaglandin release in human uterine smooth muscle cells, inhibits thus the Oxytocin (HY-17571)-induced uterine contraction and delays parturition in pregnant rats in labor.

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SSR126768A free base Chemical Structure

SSR126768A free base Chemical Structure

CAS No. : 785048-28-4

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SSR126768A free base Related Antibodies

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Description

SSR126768A free base is an orally active antagonist for oxytocin receptor, with Ki of 0.44 nM. SSR126768A free base is a tocolytic agent, that antagonizes the Oxytocin (HY-17571)-induced intracellular Ca2+ increase and prostaglandin release in human uterine smooth muscle cells, inhibits thus the Oxytocin (HY-17571)-induced uterine contraction and delays parturition in pregnant rats in labor[1].

Molecular Weight

604.52

Formula

C33H31Cl2N3O4
CAS No.
SMILES

O=C(N(CC)CC1=CN=CC=C1)C2=CC=C(Cl)C([C@](C3=C(N4CC5=CC=C(OC)C=C5OC)C=CC(Cl)=C3)(C)C4=O)=C2
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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SSR126768A free base Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SSR126768A785048-28-4Oxytocin ReceptorOXTRpreterm labororally activetocolyticSprague-Dawley CD ratsWistar ratsLtk cellDXB11UtSMCInhibitorinhibitorinhibit

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