2. GPCR/G Protein
  3. Protease Activated Receptor (PAR)
  4. UDM-001651

UDM-001651 is a potent, selective, and orally bioavailable protease-activated receptor 4 (PAR4) antagonist (IC50=4 nM; Kd=1.4 nM). UDM-001651 shows antiplatelet potency (IC50=25 nM) in a γ-thrombin-induced platelet-rich plasma aggregation assay (γ-Thr PRP).

For research use only. We do not sell to patients.

UDM-001651 Chemical Structure

UDM-001651 Chemical Structure

CAS No. : 1477497-01-0

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UDM-001651 Related Antibodies

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PAR1 PAR2 PAR4

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Description

UDM-001651 is a potent, selective, and orally bioavailable protease-activated receptor 4 (PAR4) antagonist (IC50=4 nM; Kd=1.4 nM). UDM-001651 shows antiplatelet potency (IC50=25 nM) in a γ-thrombin-induced platelet-rich plasma aggregation assay (γ-Thr PRP)[1].

IC50 & Target

PAR4

 

Molecular Weight

513.56

Formula

C28H23N3O5S
CAS No.
SMILES

COC1=CC(OCC2=CC=CC(OCC3=CC=CC=C3)=C2)=C4C=C(C5=CN6C(SC(OC)=N6)=N5)OC4=C1
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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UDM-001651 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

UDM-0016511477497-01-0UDM001651UDM 001651Protease Activated Receptor (PAR)Thrombin receptorsInhibitorinhibitorinhibit

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