Zuclomiphene-d₄ citrate

Cat. No.: HY-B1617AS Purity: ≥99.0%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

Zuclomiphene-d₄ (citrate) is a deuterium labeled Zuclomiphene citrate. Zuclomiphene citrate has an antiestrogenic effect and can inhibit the secretion of luteinizing hormone (LH) more than the trans isomer. Zuclomiphene citrate is also an orally active hypocholesterolemic agent[1][2][3][4].

For research use only. We do not sell to patients.

Zuclomiphene-d<sub>4</sub> citrate Chemical Structure

Zuclomiphene-d₄ citrate Chemical Structure

CAS No. : 2714316-71-7

Size	Price	Stock	Quantity
1 mg	USD 330	In-stock	Estimated Time of Arrival: December 31
5 mg	USD 1000	In-stock	Estimated Time of Arrival: December 31
10 mg		Get quote
50 mg		Get quote

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This product is a controlled substance and not for sale in your territory.

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Based on 1 publication(s) in Google Scholar

Other Forms of Zuclomiphene-d₄ citrate:

Zuclomiphene Get quote
Zuclomiphene citrate Get quote

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Biological Activity
Purity & Documentation
References
Customer Review

Description

Molecular Weight

602.11

Formula

C₃₂H₃₂D₄ClNO₈

CAS No.

2714316-71-7

Unlabeled CAS

7619-53-6

Appearance

Solid

Color

White to off-white

SMILES

Cl/C(C1=CC=CC=C1)=C(C2=CC=C(OC([2H])([2H])C([2H])([2H])N(CC)CC)C=C2)/C3=CC=CC=C3.O=C(CC(C(O)=O)(O)CC(O)=O)O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

DMSO : 100 mg/mL (166.08 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	1.6608 mL	8.3041 mL	16.6083 mL
5 mM	0.3322 mL	1.6608 mL	3.3217 mL
10 mM	0.1661 mL	0.8304 mL	1.6608 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)

Volume _(start)

Concentration _(final)

Volume _(final)

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
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Dosing volume
(per animal)

μL

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: ≥99.0%

Select Batch:

Data Sheet (277 KB) SDS (251 KB)

COA (257 KB) HNMR (140 KB) LCMS (87 KB)

Handling Instructions (2659 KB)

References

[1]. Fontenot GK, et al. Differential effects of isomers of clomiphene citrate on reproductive tissues in male mice. BJU Int. 2016 Feb;117(2):344-50. [Content Brief]

[2]. Mikkelson TJ, et al. Single-dose pharmacokinetics of clomiphene citrate in normal volunteers. Fertil Steril. 1986 Sep;46(3):392-6. [Content Brief]

[3]. Sutherland RL. Estrogen antagonists in chick oviduct: antagonist activity of eight synthetic triphenylethylene derivatives and their interactions with cytoplasmic and nuclear estrogen receptors. Endocrinology. 1981 Dec;109(6):2061-8. [Content Brief]

[4]. Ramsey RB, et al. The biochemical and morphological response of hydrolytic enzymes in the developing brain to hypocholesterolemic agents. Acta Neuropathol. 1980;49(2):89-94. [Content Brief]

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO / DMSO	1 mM	1.6608 mL	8.3041 mL	16.6083 mL	41.5207 mL
	5 mM	0.3322 mL	1.6608 mL	3.3217 mL	8.3041 mL
	10 mM	0.1661 mL	0.8304 mL	1.6608 mL	4.1521 mL
	15 mM	0.1107 mL	0.5536 mL	1.1072 mL	2.7680 mL
	20 mM	0.0830 mL	0.4152 mL	0.8304 mL	2.0760 mL
	25 mM	0.0664 mL	0.3322 mL	0.6643 mL	1.6608 mL
	30 mM	0.0554 mL	0.2768 mL	0.5536 mL	1.3840 mL
	40 mM	0.0415 mL	0.2076 mL	0.4152 mL	1.0380 mL
	50 mM	0.0332 mL	0.1661 mL	0.3322 mL	0.8304 mL
	60 mM	0.0277 mL	0.1384 mL	0.2768 mL	0.6920 mL
	80 mM	0.0208 mL	0.1038 mL	0.2076 mL	0.5190 mL
	100 mM	0.0166 mL	0.0830 mL	0.1661 mL	0.4152 mL