2. GPCR/G Protein
  3. Vasopressin Receptor
  4. Argipressin

Argipressin  (Synonyms: Arg8-vasopressin; AVP)

Cat. No.: HY-P0049 Purity: 99.82%
COA Handling Instructions

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Argipressin (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

Argipressin Chemical Structure

Argipressin Chemical Structure

CAS No. : 113-79-1

Size Price Stock Quantity
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in Water
ready for reconstitution
 USD 189 In-stock
Solution
10 mM * 1 mL in Water USD 189 In-stock
Solid
1 mg USD 66 In-stock
5 mg USD 119 In-stock
10 mg USD 158 In-stock
25 mg USD 211 In-stock
50 mg USD 251 In-stock
100 mg   Get quote  
200 mg   Get quote  

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Based on 12 publication(s) in Google Scholar

Other Forms of Argipressin:

Argipressin Related Antibodies

Top Publications Citing Use of Products

View All Vasopressin Receptor Isoform Specific Products:

View All Isoforms
V1a Receptor  V1b Receptor  V2 Receptor 

  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

Argipressin (Arg8-vasopressin) binds to the V1, V2, V3-vascular arginine vasopressin receptor, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells for V1.

IC50 & Target

V2 Receptor 

 

In Vitro

Argipressin binds to the vascular arginine vasopressin receptor, V1, with a Kd value of 1.31 nM in A7r5 rat aortic smooth muscle cells. It also stimulates the intracellular release of calcium in A7r5 cells (EC50=5 nM)[1]. AVP-induced [Ca2+]i signals and immunized activity against S-100 in DRG cell culture. The minimum effective concentrations of Argipressin causing [Ca2+]i responses are 100 pM in non-neuronal cells in DRG culture[2].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Argipressin Related Antibodies
Clinical Trial
Molecular Weight

1084.23

Formula

C46H65N15O12S2
CAS No.
Appearance

Solid

Color

White to off-white

Sequence

Cys-Tyr-Phe-Gln-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge: Cys1-Cys6)
Sequence Shortening

CYFQNCPRG-NH2 (Disulfide bridge: Cys1-Cys6)
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Sealed storage, away from moisture and light, under nitrogen

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 1 year; -20°C, 6 months (sealed storage, away from moisture and light, under nitrogen)

Solvent & Solubility
In Vitro: 

H2O : 100 mg/mL (92.23 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 0.9223 mL 4.6116 mL 9.2231 mL
5 mM 0.1845 mL 0.9223 mL 1.8446 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 1 year; -20°C, 6 months (sealed storage, away from moisture and light, under nitrogen). When stored at -80°C, please use it within 1 year. When stored at -20°C, please use it within 6 months.

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
This product has good water solubility, please refer to the measured solubility data in water/PBS/Saline for details.
The concentration of the stock solution you require exceeds the measured solubility. The following solution is for reference only.If necessary, please contact MedChemExpress (MCE).
Purity & Documentation

Purity: 99.82%

COA (260 KB) LCMS (86 KB) Elemental Analysis Report (119 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 1 year; -20°C, 6 months (sealed storage, away from moisture and light, under nitrogen). When stored at -80°C, please use it within 1 year. When stored at -20°C, please use it within 6 months.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
H2O 1 mM 0.9223 mL 4.6116 mL 9.2231 mL 23.0578 mL
5 mM 0.1845 mL 0.9223 mL 1.8446 mL 4.6116 mL
10 mM 0.0922 mL 0.4612 mL 0.9223 mL 2.3058 mL
15 mM 0.0615 mL 0.3074 mL 0.6149 mL 1.5372 mL
20 mM 0.0461 mL 0.2306 mL 0.4612 mL 1.1529 mL
25 mM 0.0369 mL 0.1845 mL 0.3689 mL 0.9223 mL
30 mM 0.0307 mL 0.1537 mL 0.3074 mL 0.7686 mL
40 mM 0.0231 mL 0.1153 mL 0.2306 mL 0.5764 mL
50 mM 0.0184 mL 0.0922 mL 0.1845 mL 0.4612 mL
60 mM 0.0154 mL 0.0769 mL 0.1537 mL 0.3843 mL
80 mM 0.0115 mL 0.0576 mL 0.1153 mL 0.2882 mL

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

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Argipressin Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Argipressin113-79-1Arg8-vasopressin AVPVasopressin ReceptorInhibitorinhibitorinhibit

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