1. GPCR/G Protein Neuronal Signaling
  2. Dopamine Receptor
  3. Haloperidol-d4-1

Haloperidol-d4-1 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist.

For research use only. We do not sell to patients.

Haloperidol-d<sub>4</sub>-1 Chemical Structure

Haloperidol-d4-1 Chemical Structure

CAS No. : 136765-35-0

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1 mg USD 320 In-stock
5 mg USD 800 In-stock
10 mg USD 1450 In-stock
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Based on 1 publication(s) in Google Scholar

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Description

Haloperidol-d4-1 is deuterium labeled haloperidol, and the latter is a potent dopamine D2 receptor antagonist.

IC50 & Target

D2 Receptor

 

Molecular Weight

379.89

Formula

C21H19D4ClFNO2

CAS No.
Unlabeled CAS

52-86-8

Appearance

Solid

Color

White to off-white

SMILES

OC1(CCN(CCCC(C2=C([2H])C([2H])=C(F)C([2H])=C2[2H])=O)CC1)C3=CC=C(Cl)C=C3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (263.23 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

DMSO : 100 mg/mL (263.23 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.6323 mL 13.1617 mL 26.3234 mL
5 mM 0.5265 mL 2.6323 mL 5.2647 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

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Volume (start)

V1

=
Concentration (final)

C2

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Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO / DMSO 1 mM 2.6323 mL 13.1617 mL 26.3234 mL 65.8085 mL
5 mM 0.5265 mL 2.6323 mL 5.2647 mL 13.1617 mL
10 mM 0.2632 mL 1.3162 mL 2.6323 mL 6.5809 mL
15 mM 0.1755 mL 0.8774 mL 1.7549 mL 4.3872 mL
20 mM 0.1316 mL 0.6581 mL 1.3162 mL 3.2904 mL
25 mM 0.1053 mL 0.5265 mL 1.0529 mL 2.6323 mL
30 mM 0.0877 mL 0.4387 mL 0.8774 mL 2.1936 mL
40 mM 0.0658 mL 0.3290 mL 0.6581 mL 1.6452 mL
50 mM 0.0526 mL 0.2632 mL 0.5265 mL 1.3162 mL
60 mM 0.0439 mL 0.2194 mL 0.4387 mL 1.0968 mL
80 mM 0.0329 mL 0.1645 mL 0.3290 mL 0.8226 mL
100 mM 0.0263 mL 0.1316 mL 0.2632 mL 0.6581 mL
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Product Name:
Haloperidol-d4-1
Cat. No.:
HY-14538S1
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