2. Signaling Pathways
  3. Metabolic Enzyme/Protease
  4. Carboxypeptidase
  5. Carboxypeptidase Inhibitor

Carboxypeptidase Inhibitor

Carboxypeptidase Inhibitors (11):

Cat. No. Product Name Effect Purity
  • HY-100788
    2-PMPA
    		Inhibitor ≥98.0%
    2-PMPA is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM.
  • HY-103345
    2-MPPA
    		Inhibitor ≥98.0%
    2-MPPA (GPI-5693) is an orally active and selective glutamate carboxypeptidase II (GCP II; PSMA) inhibitor with an IC50 of 90 nM.
  • HY-W044764
    2-Benzylsuccinic acid
    		Inhibitor 99.41%
    2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is an potent inhibitor of carboxypeptidase A (CPA).
  • HY-W096171
    D-Dopa
    		Inhibitor
    D-Dopa is a non-competitive, allosteric inhibitor for glutamate carboxypeptidase II (GCPII) with an IC50 of 200 nM. D-Dopa exhibits good pharmacokinetic characteristics, and low blood-brain barrier permeability in mouse model.
  • HY-70005
    CPA inhibitor
    		Inhibitor 99.93%
    CPA inhibitor (Carboxypeptidase inhibitor; compound 5) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.
  • HY-122369
    Histargin
    		Inhibitor
    Histargin is a carboxypeptidase B inhibitor with IC50 of 17 μg/ml and ＞ 100 μg/ml aganist Carboxypeptidase B and Carboxypeptidase A, respectively. Histargin can be produced by actinomycetes.
  • HY-139840A
    GCPII-IN-1 TFA
    		Inhibitor 99.99%
    GCPII-IN-1 TFA is a glutamate carboxypeptidase II (GCPII, or PSMA) inhibitor scaffold with a Ki of 44.3 nM.
  • HY-W704574
    Mergetpa
    		Inhibitor
    Mergetpa is a carboxypeptidase inhibitor used to block the conversion of kinins and B2 receptor antagonists to metabolites lacking the C-terminal arginine.
  • HY-70003
    Carboxypeptidase G2 (CPG2) Inhibitor
    		Inhibitor 98.03%
    Carboxypeptidase G2 (CPG2) Inhibitor is a novel Carboxypeptidase G2 (CPG2) Inhibitor, Antitumor agents.
  • HY-100788C
    2-PMPA sodium
    		Inhibitor
    2-PMPA sodium is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) with an IC50 of 300 pM.
  • HY-139840
    GCPII-IN-1
    		Inhibitor 99.83%
    GCPII-IN-1 is a glutamate carboxypeptidase II (GCPII, or PSMA) inhibitor scaffold with a Ki of 44.3 nM.