MAP4K Inhibitors

MAP4K2/GCK

MAP4K3/GLK

MAP4K4/HGK

MAP4K5/KHS1

MAP4K6/MINK1

MAP4K7/TNIK

MAP4K1/HPK1

MAP4K Inhibitors

Product Name	MAP4K2/GCK	MAP4K3/GLK	MAP4K4/HGK	MAP4K5/KHS1	MAP4K6/MINK1	MAP4K7/TNIK	MAP4K1/HPK1	Purity
NCB-0846						TNIK, IC₅₀: 21 nM		99.61%
GNE-495			MAP4K4, IC₅₀: 3.7 nM					99.40%
DMX-5804	GCK/MAP4K2, pIC₅₀: 6.50	GLK/MAP4K3, pIC₅₀: 4.95	MAP4K4, IC₅₀: 3 nM MAP4K4, pIC₅₀: 8.55	KHS/MAP4K5, pIC₅₀: 6.36	MINK1/MAP4K6, pIC₅₀: 8.18	TNIK/MAP4K7, pIC₅₀: 7.96		99.83%
NG25	MAP4K2, IC₅₀: 21.7 nM							99.35%
PF-06260933			MAP4K4, IC₅₀: 3.7 nM					99.67%
HPK1-IN-3							HPK1, IC₅₀: 0.25 nM	99.32%
KY-05009						TNIK, Ki: 100 nM		99.24%
HPK1-IN-7		GLK/MAP4K3, IC₅₀: 140 nM					HPK1, IC₅₀: 2.6 nM	99.33%
DS21150768							HPK1	99.26%
HPK1-IN-32							HPK1	98.12%
ZYF0033							HPK1, IC₅₀: <10 nM	98.86%
MAP4K4-IN-3			MAP4K4, IC₅₀: 14.9 nM					99.15%
GNE 220 hydrochloride			MAP4K4, IC₅₀: 7 nM	MAP4K5, IC₅₀: 9 nM	MAP4K6, IC₅₀: 1.1 μM			98.22%
INS018 055			MAP4K4, IC₅₀: 12-120 nM					99.38%
TAK1/MAP4K2 inhibitor 1	MAP4K2, IC₅₀: 18.2 nM							99.90%
HPK1-IN-26							HPK1	≥98.0%
HPK1-IN-34							HPK1, IC₅₀: <100 nM
DB1113	MAP4K2	GLK/MAP4K3		MAP4K5			HPK1	99.28%
GNE-6893							HPK1	99.94%
SS47							HPK1
GNE 220			MAP4K4, IC₅₀: 7 nM	MAP4K5, IC₅₀: 9 nM	MAP4K6, IC₅₀: 1.1 μM
HPK1-IN-21							HPK1, Ki: 0.8 nM
HPK1-IN-36							HPK1, IC₅₀: 0.5 nM
RET-IN-19			MAP4K4, IC₅₀: 3.428 ± 0. μM
FLT3/ITD-IN-4			MAP4K4, EC₅₀: 5737 nM
HPK1-IN-44							HPK1, IC₅₀: 0.1 nM
HPK1-IN-35							HPK1, IC₅₀: 3.5 nM
HPK1-IN-49							HPK1
HPK1-IN-52	MAP4K2, IC₅₀: 448 nM	GLK/MAP4K3, IC₅₀: 85 nM	MAP4K4, IC₅₀: 665 nM	MAP4K5, IC₅₀: 104 nM	MAP4K6, IC₅₀: 168 nM		HPK1, IC₅₀: 10.4 nM
HPK1-IN-24							HPK1, Ki: <100 nM
HPK1-IN-25							HPK1, IC₅₀: 129 nM
HPK1-IN-33							HPK1, Ki: 1.7 nM
KHK-6							HPK1, IC₅₀: 20 nM
HPK1-IN-43							HPK1, IC₅₀: 0.32 nM

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