PAK Inhibitors

PAK1

PAK2

PAK3

PAK4

PAK5

PAK6

PAK Inhibitors & Activators

Product Name	PAK1	PAK2	PAK3	PAK4	PAK5	PAK6	Purity
Fingolimod hydrochloride	PAK1						99.95%
5-Aminosalicylic Acid	PAK1						99.82%
Fingolimod	PAK1						99.97%
PF-3758309	PAK1, Ki: 13.7 nM	PAK2, IC₅₀: 190 nM	PAK3, IC₅₀: 99 nM	PAK4, Ki: 18.7 nM PAK4, Kd: 2.7 nM	PAK5, Ki: 18.1 nM	PAK6, Ki: 17.1 nM	99.84%
IPA-3	PAK1, IC₅₀: 2.5 μM						99.43%
PAK4-IN-5	PAK1, IC₅₀: 1872.01 nM			PAK4, IC₅₀: 7.68 nM
FRAX597	PAK1, IC₅₀: 8 nM	PAK2, IC₅₀: 13 nM	PAK3, IC₅₀: 19 nM				99.79%
PRT062607 Hydrochloride					PAK5, IC₅₀: 166 nM (^[2])		98.07%
FRAX486	PAK1, IC₅₀: 14 nM	PAK2, IC₅₀: 33 nM	PAK3, IC₅₀: 39 nM				98.01%
G-5555	PAK1, Ki: 3.7 nM	PAK2, Ki: 11 nM					99.88%
Padnarsertib				PAK4, IC₅₀: 100 nM			99.86%
FRAX1036	PAK1, Ki: 23.3 nM	PAK2, Ki: 72.4 nM		PAK4, Ki: 2.4 μM			99.49%
AZ13705339	PAK1, Kd: 0.28 nM PAK1, IC₅₀: 0.33 nM pPAK1, IC₅₀: 59 nM	PAK2, Kd: 0.32 nM					98.90%
LCH-7749944				PAK4, IC₅₀: 14.93 μM			99.36%
G-5555 hydrochloride	PAK1, Ki: 3.7 nM	PAK2, Ki: 11 nM					98.78%
PAK4-IN-2			PAK3, IC₅₀: 2.7 nM				99.78%
NVS-PAK1-C	PAK1, Kd: 0.007 μM PAK1, IC₅₀: 5 nM	PAK2, Kd: 0.4 μM PAK2, IC₅₀: 270 nM					≥99.0%
PRT062607 acetate					PAK5, IC₅₀: 166 nM (^[2])		99.83%
AZ13705339 hemihydrate	PAK1, Kd: 0.28 nM PAK1, IC₅₀: 0.33 nM pPAK1, IC₅₀: 59 nM	PAK2, Kd: 0.32 nM					99.77%
PAK1-IN-1	PAK1, IC₅₀: 9.8 nM			PAK4, IC₅₀: >10 μM
PF-3758309 hydrochloride	PAK1, Ki: 13.7 nM	PAK2, IC₅₀: 190 nM	PAK3, IC₅₀: 99 nM	PAK4, Ki: 18.7 nM PAK4, Kd: 2.7 nM	PAK5, Ki: 18.1 nM	PAK6, Ki: 17.1 nM
PF-3758309 dihydrochloride	PAK1, Ki: 13.7 nM	PAK2, IC₅₀: 190 nM	PAK3, IC₅₀: 99 nM	PAK4, Ki: 18.7 nM PAK4, Kd: 2.7 nM	PAK5, Ki: 18.1 nM	PAK6, Ki: 17.1 nM
G-9791	PAK1, Ki: 0.95 nM	PAK2, Ki: 2.0 nM
2,2′-Dihydroxy-6,6′-dinaphthyl disulfide	PAK1
Mesalamine impurity P	PAK1
PAK4-IN-1				PAK4
ZINC194100678	PAK1, IC₅₀: 8.37 μM
ZMF-10	PAK1, IC₅₀: 174 nM	PAK2, IC₅₀: 1.038 μM	PAK3, IC₅₀: 1.372 μM
KY-04045				PAK4, IC₅₀: 8.7 μM
AK963/40708899	PAK1

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