2. Cell Cycle/DNA Damage Cytoskeleton
  3. PAK
  4. G-9791

G-9791, a poyridone side chain analogue, is a potent PAK inhibitor with Ki values of 0.95 nM and 2.0 nM for PAK1 and PAK2, respectively.

For research use only. We do not sell to patients.

G-9791 Chemical Structure

G-9791 Chemical Structure

CAS No. : 1926204-95-6

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G-9791 Related Antibodies

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Description

G-9791, a poyridone side chain analogue, is a potent PAK inhibitor with Ki values of 0.95 nM and 2.0 nM for PAK1 and PAK2, respectively[1].

IC50 & Target[1]

PAK1

0.95 nM (Ki)

PAK2

2.0 nM (Ki)

Molecular Weight

508.98

Formula

C26H26ClFN6O2
CAS No.
SMILES

O=C1C(C2=CC=C(N3C=CC=C(C)C3=O)C=C2Cl)=CC4=CN=C(NC)N=C4N1CCC5(F)CN(C)C5
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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G-9791 Related Classifications

  • Molarity Calculator

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

G-97911926204-95-6G9791G 9791PAKp21 activated kinasespoyridone side chainInhibitorinhibitorinhibit

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HY-116917
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