1. Signaling Pathways
  2. Stem Cell/Wnt
    TGF-beta/Smad
  3. PKA
  4. PKA Inhibitors

PKA Inhibitors

PKA

PKAR

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PKA Inhibitors, Agonists & Activators
Product Name PKA PKAR Purity
Bucladesine sodium
PKA
  99.48%
Fasudil Hydrochloride
PKA, IC50: 4.58 μM
  99.96%
Daphnetin
PKA, IC50: 9.33 μM
  99.86%
Bucladesine calcium
PKA
  99.52%
PKA Inhibitor Fragment (6-22) amide TFA
PKA, Ki: 2.8 nM
  99.77%
AT7867
PKA, IC50: 20 nM
  99.88%
KT5823
PKA, Ki: 10 μM
  99.90%
AT13148
PKA, IC50: 3 nM
  99.21%
Bilobetin
PKA
  99.39%
AT7867 dihydrochloride
PKA, IC50: 20 nM
  99.75%
CW 008
PKA
  98.15%
Sp-cAMPS sodium salt
PKA I
PKA II
  99.45%
Jaspamycin
Trypanosoma brucei PKA holoenzyme, Kd: 8 nM
Trypanosoma brucei PKAR(199-499), EC50: 6.5 nM
98.60%
Sp-cAMPS
PKA I
PKA II
 
A-3 hydrochloride
PKA, Ki: 4.3 μM
  99.75%
Hu7691
PKA, IC50: 11 nM
 
Akt1&PKA-IN-1
PKAa, IC50: 0.03 μM
 
Fasudil
PKA, IC50: 4.58 μM
 
Hu7691 free base
PKA, IC50: 11 nM
 
Fasudil dihydrochloride
PKA, IC50: 4.58 μM
 
Fasudil hydrochloride semihydrate
PKA, IC50: 4.58 μM
 
Sp-cAMPS triethylamine
PKA I
PKA II
 
Sp-8-Br-cAMPS sodium
PKA, EC50: 360 nM
 
PKA Inhibitor Fragment (6-22) amide
PKA, Ki: 2.8 nM
 
HA-100 hydrochloride
PKA, IC50: 8 μM
 
HA-100 dihydrochloride
PKA, IC50: 8 μM
 
GSK466317A
PKA, IC50: 12.59 μM
 
PF-4950834
PKA, IC50: 424 nM
 
Balanol
PKA
 
LX7101 monohydrochloride
PKA, IC50: <1 nM