1. Signaling Pathways
  2. Immunology/Inflammation
  3. SphK
  4. SphK Inhibitors

SphK Inhibitors

SphK1

SphK2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

SphK Inhibitors & Activators
Product Name SphK1 SphK2 Purity
PF-543
SphK1
  99.85%
PF-543 Citrate
SphK1
  99.47%
RB-005
SphK1, IC50: 3.6 μM
 
K145 hydrochloride  
SphK2
99.88%
K6PC-5
SphK1
  99.85%
SKI-178
SphK1
SphK2
98.91%
MHP
SphK1
  98.23%
MP-A08
SphK1
  ≥98.0%
Amgen-23
SphK1, IC50: 20 nM
SphK2, IC50: 1.6 μM
99.00%
SK1-​I hydrochloride
SphK1
  99.49%
SphK1&2-IN-1
SphK1
SphK2
99.33%
SphK1-IN-2
SphK1, IC50: 19.81 nM
SphK2, IC50: >10 μM
SphK2-IN-1  
SphK2, IC50: 0.359 μM
SphK1-IN-1
SphK1
 
SphK1-IN-3
SphK1, IC50: 2.48 μM