1. Signaling Pathways
  2. Immunology/Inflammation
  3. IKZF Family
  4. IKZF Family Inhibitors

IKZF Family Inhibitors

IKZF1

IKZF2

IKZF3

IKZF4

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

IKZF Family Degraders & Inhibitors
Product Name IKZF1 IKZF2 IKZF3 IKZF4 Purity
NVP-DKY709  
IZKF2, DC50: 4 nM
 
IKZF4, DC50: 13 nM
98.86%
Cemsidomide
IKZF1
 
IKZF3
  99.54%
ALV1
IKZF1, DC50: 2.5 nM
IZKF2, DC50: 10.3 nM
    98.62%
MGD-4
IKZF1, DC50: 67.2 nM
IZKF2, DC50: 918.2 nM
IKZF3, DC50: 95.8 nM
 
BMS-986449  
IKZF2
 
IKZF4
MG degrader 1    
IKZF3, EC50: 1.385 nM
  99.83%
IKZF3 degrader 1    
IKZF3, EC50: 0.012 μM
 
MGD-28
IKZF1, DC50: 3.8 nM
IZKF2, DC50: 56.3 nM
IKZF3, DC50: 7.1 nM
 
IKZF1-degrader-1
IKZF1, DC50: 0.134 nM