Anticancer agent 230

Cat. No.: HY-164064 Purity: 99.97%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

Anticancer agent 230 (example 65) is a caseinolytic protease P (ClpP) activator with anticancer activity. Anticancer agent 230 is able to induce the degradation of mitochondrial proteins in SUM159 and MDA-MB-231 triple-negative breast cancer cells in a time-dependent manner.

For research use only. We do not sell to patients.

Anticancer agent 230 Chemical Structure

CAS No. : 2485052-87-5

Size	Price	Stock	Quantity
5 mg	USD 50	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 80	In-stock	Estimated Time of Arrival: December 31
25 mg	USD 160	In-stock	Estimated Time of Arrival: December 31
50 mg	USD 255	In-stock	Estimated Time of Arrival: December 31
100 mg	USD 400	Get quote	Estimated Time of Arrival: December 31
200 mg		Get quote
500 mg		Get quote

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Based on 1 publication(s) in Google Scholar

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Purity & Documentation
References
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Description

Molecular Weight

390.87

Formula

C₂₂H₁₉ClN₄O

CAS No.

2485052-87-5

Appearance

Solid

Color

White to off-white

SMILES

N#CC1=CC=CC(CN(C2)CCC(N=CN3CC4=CC=C(Cl)C=C4)=C2C3=O)=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

Solvent & Solubility

In Vitro:

DMSO : 50 mg/mL (127.92 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.5584 mL	12.7920 mL	25.5840 mL
5 mM	0.5117 mL	2.5584 mL	5.1168 mL
10 mM	0.2558 mL	1.2792 mL	2.5584 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)

Volume _(start)

Concentration _(final)

Volume _(final)

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

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μL

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: 99.97%

Select Batch:

Data Sheet (267 KB) SDS (251 KB)

COA (244 KB) HNMR (241 KB) RP-HPLC (266 KB) LCMS (95 KB)

Handling Instructions (2659 KB)

References

[1]. Preparation of tetrahydropyrido[4,3-d]pyrimidine-2,4-dione analogs useful in the treatment of cancers and in modulating the activity of caseinolytic protease p function. United States, US20230339947 A1. 2023-10-26.

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	2.5584 mL	12.7920 mL	25.5840 mL	63.9599 mL
	5 mM	0.5117 mL	2.5584 mL	5.1168 mL	12.7920 mL
	10 mM	0.2558 mL	1.2792 mL	2.5584 mL	6.3960 mL
	15 mM	0.1706 mL	0.8528 mL	1.7056 mL	4.2640 mL
	20 mM	0.1279 mL	0.6396 mL	1.2792 mL	3.1980 mL
	25 mM	0.1023 mL	0.5117 mL	1.0234 mL	2.5584 mL
	30 mM	0.0853 mL	0.4264 mL	0.8528 mL	2.1320 mL
	40 mM	0.0640 mL	0.3198 mL	0.6396 mL	1.5990 mL
	50 mM	0.0512 mL	0.2558 mL	0.5117 mL	1.2792 mL
	60 mM	0.0426 mL	0.2132 mL	0.4264 mL	1.0660 mL
	80 mM	0.0320 mL	0.1599 mL	0.3198 mL	0.7995 mL
	100 mM	0.0256 mL	0.1279 mL	0.2558 mL	0.6396 mL