2. Metabolic Enzyme/Protease
  3. Phosphatase
  4. CaMKP inhibitor sodium

CaMKP inhibitor sodium (compound 5) is an inhibitor of Ca2+/neutral protein-dependent protein concentration (CaMKP) and its nuclear type (CaMKP-N) (IC50: 6.4 μM, CaMKP; 6.6 μM, CaMKP-N). CaMKP is one type of Ser/Thr protein, which can be passed through to remove the oxidized oxidized protein (CaMK). CaMKP inhibitor sodium inhibits CaMKP mediated phospho-CaMKI hydrolysis, unaffectes protein phosphoric acid 2C (PP2C) and calcineurin (CaN).

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CaMKP inhibitor sodium Chemical Structure

CaMKP inhibitor sodium Chemical Structure

CAS No. : 52789-62-5

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CaMKP inhibitor sodium Related Antibodies

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Description

CaMKP inhibitor sodium (compound 5) is an inhibitor of Ca2+/neutral protein-dependent protein concentration (CaMKP) and its nuclear type (CaMKP-N) (IC50: 6.4 μM, CaMKP; 6.6 μM, CaMKP-N). CaMKP is one type of Ser/Thr protein, which can be passed through to remove the oxidized oxidized protein (CaMK). CaMKP inhibitor sodium inhibits CaMKP mediated phospho-CaMKI hydrolysis, unaffectes protein phosphoric acid 2C (PP2C) and calcineurin (CaN)[1].

IC50 & Target

IC50: 6.4 μM (CaMKP); 6.6 μM (CaMKP-N)[1]
In Vitro

CaMKP inhibitor sodium (10 μM; 6 h) inhibits CaMKP-N expressed in Neuro2a cells[1].
CaMKP inhibitor sodium (2.5 μM, 5 μM) inhibits CaMKP activity instead of PP2C activity in Neuro2a cells[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

CaMKP inhibitor sodium Related Antibodies
Molecular Weight

341.29

Formula

C10H8NNaO7S2
CAS No.
Appearance

Solid

Color

Gray to brown

SMILES

O=S(C1=C2C=CC=C(O)C2=C(N)C(S(=O)(O)=O)=C1)(O[Na])=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Solvent & Solubility
In Vitro: 

DMSO : 5 mg/mL (14.65 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.9301 mL 14.6503 mL 29.3006 mL
5 mM 0.5860 mL 2.9301 mL 5.8601 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.9301 mL 14.6503 mL 29.3006 mL 73.2515 mL
5 mM 0.5860 mL 2.9301 mL 5.8601 mL 14.6503 mL
10 mM 0.2930 mL 1.4650 mL 2.9301 mL 7.3251 mL
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CaMKP inhibitor sodium Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CaMKP inhibitor52789-62-5PhosphataseInhibitorinhibitorinhibit

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