EST64454 maleate

Cat. No.: HY-131914B: Data Sheet Handling Instructions Technical Support

EST64454 maleate is a highly soluble σ1 receptor antagonist, demonstrating potent antinociceptive properties for pain treatment. EST64454 maleate exhibits excellent metabolic stability across various species and possesses an adequate pharmacokinetic profile in rodents. EST64454 maleate has been identified as a promising clinical candidate due to its favorable aqueous solubility and high permeability in Caco-2 cells.

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EST64454 maleate Chemical Structure

CAS No. : 2088272-67-5

Size	Price	Stock	Quantity
1 mg	USD 215	Get quote 3 - 4 weeks 2 - 3 weeks 2 - 3 weeks	2 - 3 weeks
5 mg	USD 481	Get quote 3 - 4 weeks 2 - 3 weeks 2 - 3 weeks	2 - 3 weeks
10 mg	USD 712	Get quote 3 - 4 weeks 2 - 3 weeks 2 - 3 weeks	2 - 3 weeks
25 mg	USD 1133	Get quote 3 - 4 weeks 2 - 3 weeks 2 - 3 weeks	2 - 3 weeks
50 mg	USD 1537	Get quote 3 - 4 weeks 2 - 3 weeks 2 - 3 weeks	2 - 3 weeks
100 mg		Get quote
200 mg		Get quote

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Based on 1 publication(s) in Google Scholar

Other Forms of EST64454 maleate:

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Purity & Documentation
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Description	EST64454 maleate is a highly soluble σ1 receptor antagonist, demonstrating potent antinociceptive properties for pain treatment. EST64454 maleate exhibits excellent metabolic stability across various species and possesses an adequate pharmacokinetic profile in rodents. EST64454 maleate has been identified as a promising clinical candidate due to its favorable aqueous solubility and high permeability in Caco-2 cells.
Molecular Weight	480.46
Formula	C₂₂H₂₆F₂N₄O₆
CAS No.	2088272-67-5
SMILES	OC(/C=C\C(O)=O)=O.CC(N(CC1)CCN1CCOCC2=NN(C3=CC(F)=C(C=C3)F)C=C2)=O
Shipping	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation	Data Sheet (266 KB) Handling Instructions (2659 KB)
References	[1]. EST64454: a Highly Soluble σ1 Receptor Antagonist Clinical Candidate for Pain Management [Content Brief]