2. Immunology/Inflammation
  3. PSMA
  4. MIP-1095 TFA

MIP-1095 TFA  (Synonyms: RPS-001 TFA)

Cat. No.: HY-123733A Purity: 99.76%
Data Sheet
SDS
COA
Handling Instructions Technical Support

Solubility

In Vivo Dissolution Calculator

MIP-1095 (RPS-001) TFA is a potent inhibitor of PSMA with good biodistribution and efficient targeting of tumor lesions. In applications, MIP-1095 TFA will be isotopically labeled (131I labeled) as an imaging probe to indicate tumor progression. And 131I-MIP-1095 showed higher renal uptake in mice.

For research use only. We do not sell to patients.

MIP-1095 TFA Chemical Structure

MIP-1095 TFA Chemical Structure

Size Price Stock Quantity
5 mg USD 225 In-stock
10 mg USD 360 In-stock
25 mg USD 720 In-stock
50 mg USD 1150 In-stock
100 mg   Get quote  
200 mg   Get quote  

Get it by April 25 for select sizes. Order within 19 hrs 58 mins.

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Based on 1 publication(s) in Google Scholar

Other Forms of MIP-1095 TFA:

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Description

MIP-1095 (RPS-001) TFA is a potent inhibitor of PSMA with good biodistribution and efficient targeting of tumor lesions. In applications, MIP-1095 TFA will be isotopically labeled (131I labeled) as an imaging probe to indicate tumor progression. And 131I-MIP-1095 showed higher renal uptake in mice[1][2].

Molecular Weight

678.35

Formula

C21H26F3IN4O10
Appearance

Solid

Color

White to off-white

SMILES

O=C([C@H](CCC(O)=O)NC(N[C@@H](CCCCNC(NC1=CC=C(C=C1)I)=O)C(O)=O)=O)O.OC(C(F)(F)F)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Solvent & Solubility
In Vitro: 

DMSO : 125 mg/mL (184.27 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.4742 mL 7.3708 mL 14.7417 mL
5 mM 0.2948 mL 1.4742 mL 2.9483 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 1.4742 mL 7.3708 mL 14.7417 mL 36.8541 mL
5 mM 0.2948 mL 1.4742 mL 2.9483 mL 7.3708 mL
10 mM 0.1474 mL 0.7371 mL 1.4742 mL 3.6854 mL
15 mM 0.0983 mL 0.4914 mL 0.9828 mL 2.4569 mL
20 mM 0.0737 mL 0.3685 mL 0.7371 mL 1.8427 mL
25 mM 0.0590 mL 0.2948 mL 0.5897 mL 1.4742 mL
30 mM 0.0491 mL 0.2457 mL 0.4914 mL 1.2285 mL
40 mM 0.0369 mL 0.1843 mL 0.3685 mL 0.9214 mL
50 mM 0.0295 mL 0.1474 mL 0.2948 mL 0.7371 mL
60 mM 0.0246 mL 0.1228 mL 0.2457 mL 0.6142 mL
80 mM 0.0184 mL 0.0921 mL 0.1843 mL 0.4607 mL
100 mM 0.0147 mL 0.0737 mL 0.1474 mL 0.3685 mL
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MIP-1095 TFA Related Classifications

Keywords:

MIP-1095RPS-001MIP1095MIP 1095RPS001RPS 001PSMAProstate-specific membrane antigenalbuminprostate cancertargeted radiotherapyInhibitorinhibitorinhibit

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