2. Epigenetics TGF-beta/Smad
  3. PKC
  4. PKCα (C2-4) inhibitor peptide

PKCα (C2-4) inhibitor peptide is a PKCα specific inhibitor peptide that blocks the inhibition of IKr by the α1A adrenoreceptor agonist A-61603 (HY-101366).

For research use only. We do not sell to patients.

Custom Peptide Synthesis

PKCα (C2-4) inhibitor peptide Chemical Structure

PKCα (C2-4) inhibitor peptide Chemical Structure

Size Price Stock Quantity
5 mg USD 85 In-stock
10 mg USD 135 In-stock
25 mg USD 270 In-stock
50 mg USD 430 In-stock
100 mg USD 650 In-stock
200 mg   Get quote  
500 mg   Get quote  

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This product is a controlled substance and not for sale in your territory.

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Based on 1 publication(s) in Google Scholar

PKCα (C2-4) inhibitor peptide Related Antibodies

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Description

PKCα (C2-4) inhibitor peptide is a PKCα specific inhibitor peptide that blocks the inhibition of IKr by the α1A adrenoreceptor agonist A-61603 (HY-101366)[1].

IC50 & Target

PKCα[1]
Molecular Weight

1107.17

Formula

C47H74N14O17
Appearance

Solid

Color

White to off-white

Sequence

Ser-Leu-Asn-Pro-Glu-Tyr-Arg-Gln-Thr
Sequence Shortening

SLNPEYRQT
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Sealed storage, away from moisture

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (90.32 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 0.9032 mL 4.5160 mL 9.0320 mL
5 mM 0.1806 mL 0.9032 mL 1.8064 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Purity: 99.81%

COA (257 KB) LCMS (106 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 0.9032 mL 4.5160 mL 9.0320 mL 22.5801 mL
5 mM 0.1806 mL 0.9032 mL 1.8064 mL 4.5160 mL
10 mM 0.0903 mL 0.4516 mL 0.9032 mL 2.2580 mL
15 mM 0.0602 mL 0.3011 mL 0.6021 mL 1.5053 mL
20 mM 0.0452 mL 0.2258 mL 0.4516 mL 1.1290 mL
25 mM 0.0361 mL 0.1806 mL 0.3613 mL 0.9032 mL
30 mM 0.0301 mL 0.1505 mL 0.3011 mL 0.7527 mL
40 mM 0.0226 mL 0.1129 mL 0.2258 mL 0.5645 mL
50 mM 0.0181 mL 0.0903 mL 0.1806 mL 0.4516 mL
60 mM 0.0151 mL 0.0753 mL 0.1505 mL 0.3763 mL
80 mM 0.0113 mL 0.0565 mL 0.1129 mL 0.2823 mL
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PKCα (C2-4) inhibitor peptide Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PKCα (C2-4) inhibitor peptidePKCProtein kinase CInhibitorinhibitorinhibit

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