2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. (±)-Penbutolol

(±)-Penbutolol  (Synonyms: (Rac)-Penbutolol; (±)-Isopenbutolol)

Cat. No.: HY-116790B
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(±)-Penbutolol ((Rac)-Penbutolol) is the racemic mixture of Penbutolol. (±)-Penbutolol is an orally active β-adrenergic receptor antagonist. (±)-Penbutolol antagonizes exercise-induced tachycardia, reduces the increase in peak expiratory flow rate (PEFR) caused by exercise, and decreases resting plasma renin activity (PRA). (±)-Penbutolol reaches peak plasma concentration 1 hour after oral administration, with a half-life of 4.5 hours, and is converted into an active metabolite in the body. (±)-Penbutolol can be used in cardiovascular-related disease research.

For research use only. We do not sell to patients.

(±)-Penbutolol Chemical Structure

(±)-Penbutolol Chemical Structure

CAS No. : 36507-48-9

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Other Forms of (±)-Penbutolol:

(±)-Penbutolol Related Antibodies

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Description

(±)-Penbutolol ((Rac)-Penbutolol) is the racemic mixture of Penbutolol. (±)-Penbutolol is an orally active β-adrenergic receptor antagonist. (±)-Penbutolol antagonizes exercise-induced tachycardia, reduces the increase in peak expiratory flow rate (PEFR) caused by exercise, and decreases resting plasma renin activity (PRA). (±)-Penbutolol reaches peak plasma concentration 1 hour after oral administration, with a half-life of 4.5 hours, and is converted into an active metabolite in the body. (±)-Penbutolol can be used in cardiovascular-related disease research[1].

IC50 & Target

Beta-1 adrenergic receptor

 

Molecular Weight

291.43

Formula

C18H29NO2
CAS No.
SMILES

OC(CNC(C)(C)C)COC1=CC=CC=C1C2CCCC2
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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(±)-Penbutolol Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

(±)-Penbutolol36507-48-9(Rac)-Penbutolol (±)-IsopenbutololAdrenergic ReceptorBeta ReceptorInhibitorinhibitorinhibit

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