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derivate

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56

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4

Fluorescent Dye

2

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12

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1

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1

Oligonucleotides

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-107784
    Ectoine

    		Bacterial Inflammation/Immunology
    Ectoine is a natural cell protectant, an amino acid derivate produced by bacteria living under extremely harsh environmental conditions. Ectoine serves as an osmoregulatory compatible solute, increasing the hydration of the skin surface and stabilizing lipid layers, which is useful in skincare. Ectoine demonstrates a good safety profile for the treatment of allergic rhinitis .
    Ectoine
  • HY-149334
    ZLD115

    		Fat Mass and Obesity-associated Protein (FTO) Metabolic Disease
    ZLD115 (compound 44) is a FB23-derivated inhibitor of Fat Mass and Obesity-associated Protein (FTO). ZLD115 is an antileukemic agent, exhibiting antiproliferative activity against leukemic cell lines .
    ZLD115
  • HY-B1345
    Piroctone olamine

    Piroctone ethanolamine

    		 Fungal Infection
    Piroctone olamine is a pyridine derivate. It is known to have a fungicidal effect.
    Piroctone olamine
  • HY-N6911A
    18α-Glycyrrhizic acid

    		Others Inflammation/Immunology
    18α-Glycyrrhizic acid is a derivate of Glycyrrhizic acid. 18α-Glycyrrhizic acid has weak antihepatotoxic anti-inflammatory activities .
    18α-Glycyrrhizic acid
  • HY-W145597
    D-Glucuronamide

    		Drug Derivative Others
    D-Glucuronamide is the derivate of D-glucuronic acid .
    D-Glucuronamide
  • HY-105191
    Azalanstat

    RS-21607

    		 Cytochrome P450 Reactive Oxygen Species Infection Inflammation/Immunology
    Azalanstat is an imidazole-dioxolane derivate that is a lanosterol 14-α demethylase inhibitor. Azalanstat is also a HO-1 (IC50 = 5.5 µM) and HO-2 (IC50 = 24.5 µM) inhibitor .
    Azalanstat
  • HY-107784R
    Ectoine (Standard)

    		Bacterial Inflammation/Immunology
    Ectoine (Standard) is the analytical standard of Ectoine. This product is intended for research and analytical applications. Ectoine is a natural cell protectant, an amino acid derivate produced by bacteria living under extremely harsh environmental conditions. Ectoine serves as an osmoregulatory compatible solute, increasing the hydration of the skin surface and stabilizing lipid layers, which is useful in skincare. Ectoine demonstrates a good safety profile for the treatment of allergic rhinitis .
    Ectoine (Standard)
  • HY-N4303
    5-​Ethoxy-​10-​Gingerol

    		Drug Derivative Others
    5-​Ethoxy-​10-​Gingerol is a derivate of gingerol.
    5-​Ethoxy-​10-​Gingerol
  • HY-N6898
    3-O-Acetylbufotalin

    		Drug Derivative Cancer
    3-O-Acetylbufotalin is a derivate of bufadienolide, with anti-cancer activity .
    3-O-Acetylbufotalin
  • HY-D1893
    HEX azide, 6-isomer

    		Fluorescent Dye Others
    HEX azide, 6-isomer, a derivate of fluorescent dye hexachlorofluorescein (HEX), can be used for labeling oligonucleotides .
    HEX azide, 6-isomer
  • HY-N1567
    Pterolactam

    		Fungal Infection
    Pterolactam can be isolated from Chrysanthemum coronarium L. Pterolactam derivates serval analogues that Mannich bases of amide with antifungal activities and cytotoxicity .
    Pterolactam
  • HY-N13187
    7,3'-Dihydroxy flavonone-4'-O-β-D-glucopyranoside

    		Others Others
    7,3'-Dihydroxy flavonone-4'-O-β-D-glucopyranoside is derivated from the seeds of Sophora alopecuroides L. .
    7,3'-Dihydroxy flavonone-4'-O-β-D-glucopyranoside
  • HY-N10017
    Lucidone F

    		Others Metabolic Disease Inflammation/Immunology
    Lucidone F is a nortriterpenoid analogue which is derivated from Ganoderma resinaceum. Lucidone F is promising for research of immune-regulation, hyperglycemia and liver disease .
    Lucidone F
  • HY-W721596
    Pentadecanoyl ethanolamide

    		Endogenous Metabolite Neurological Disease
    Pentadecanoyl ethanolamide is derivate of endougenous lipid amides, the N-acylethanolamines. Pentadecanoyl ethanolamide exhibits anticonvulsant efficacy in electroshocked mice without significant toxicity .
    Pentadecanoyl ethanolamide
  • HY-164112
    1,2-Dioleoyl-sn-glycero-3-(cytidine diphosphate) ammonium

    18:1 CDP DG

    		 Biochemical Assay Reagents Others
    1,2-Dioleoyl-sn-glycero-3-(cytidine diphosphate) ammonium (18:1 CDP DG) is a diacylglycerol derivate .
    1,2-Dioleoyl-sn-glycero-3-(cytidine diphosphate) ammonium
  • HY-B1345R
    Piroctone olamine (Standard)

    		Fungal Infection
    Piroctone olamine (Standard) is the analytical standard of Piroctone olamine. This product is intended for research and analytical applications. Piroctone olamine is a pyridine derivate. It is known to have a fungicidal effect.
    Piroctone olamine (Standard)
  • HY-W015815
    6-Methylnicotinamide

    		Endogenous Metabolite Neurological Disease
    6-Methylnicotinamide, a derivate of nicotinamide, is an endogenous metabolite. A sudden increase of 6-methylnicotinamide in the acute stages of intracerebral hemorrhage (ICH) exacerbates neurological damages .
    6-Methylnicotinamide
  • HY-N7288
    Trilepisflavan

    		Others Others
    Trilepisflavan is a flavan, which can be isolated from Trilepisium madagascariense. Trilepisflavan derivates serval analogues with anti-cancer activity against human cancer cells .
    Trilepisflavan
  • HY-N13186
    δ-(E)-Deoxy-amplexichromanol

    		Bacterial Infection
    δ-(E)-Deoxy-amplexichromanol is a δ-tocotrienolic acid derivative with potent antibacterial activities, which is derivated from hydromethanolic extract of the cones of C. atlantica .
    δ-(E)-Deoxy-amplexichromanol
  • HY-107831
    5-Acetylsalicylic acid
    1 Publications Verification

    		 Others Inflammation/Immunology
    5-Acetylsalicylic acid has anti-inflammatory and is considered to be the active agent in inflammatory bowel disease (IBD) . 5-Acetylsalicylic acid is the derivate of Acetylsalicylic acid (HY-14654).
    5-Acetylsalicylic acid
  • HY-117568
    A-80b

    		Calcium Channel Cardiovascular Disease
    A-80b is a pyridazino[4,5-b]indole derivate. A 80b showsantihypertensive activity and can be used for study of Arterial hypertension .
    A-80b
  • HY-155067
    Antitubercular agent-38

    		Bacterial Infection
    Antitubercular agent-38 is an orally active Benzothiazinones (BTZs) derivate, with potent antituberculosis activity. Antitubercular agent-38 exhibits low cardiac toxicity, low cell cytotoxicity .
    Antitubercular agent-38
  • HY-N6654
    Syringyl Alcohol

    Syringic Alcohol

    		 Drug Derivative Others
    Syringyl Alcohol (Syringic Alcohol) is a derivate of phenol comprises both phenolic and alcoholic functional groups. Syringyl Alcohol is a probe molecule for the evaluation of the catalytic performance of various carbonaceous nanomaterials (CNMs) .
    Syringyl Alcohol
  • HY-113053
    Prostaglandin A1

    		Endogenous Metabolite Apoptosis Neurological Disease Inflammation/Immunology Endocrinology Cancer
    Prostaglandin A1 is a dehydration derivate of Prostaglandin E1. Prostaglandin A1 exhibits inhibitory activities against tumor growth, inflammation, virus replication, platelet aggregation and excitotoxin-induced neurons apoptosis .
    Prostaglandin A1
  • HY-N1300
    Shizukanolide F

    		Fungal Infection Cancer
    Shizukanolide F is a dimeric sesquiterpene, which is derivated from Chloranthus japonicus Sieb. Shizukanolide F exhibits potent antifungal activities against various plant pathogenic fungi and anti-metastasis breast cancer .
    Shizukanolide F
  • HY-D0807
    5-IAF
    1 Publications Verification

    5-Iodoacetamidofluorescein

    		 Fluorescent Dye Cancer
    5-IAF (5-Iodoacetamidofluorescein) is an idoacetamide derivate of fluoresceine. 5-IAF can be used as fluorescent probe that labels proteins and other molecules having free thiols (cysteine side chains) .
    5-IAF
  • HY-107336
    Cyclovalone

    Beveno

    		 COX Inflammation/Immunology
    Cyclovalone (Beveno) is a synthetic curcumin derivate, which inihibits cyclooxygenase and exhibits anti-inflammatory, antitumor and antioxidant activities . Cyclovalone inhibits cell proliferation in normal and malignant prostatic cells. Cyclovalone ist orally active .
    Cyclovalone
  • HY-108278
    Zolimidine

    		Drug Derivative Endocrinology
    Zolimidine, a derivate of imidazopyridine, is an orally active antiulcer agent. Zolimidine stimulates mucus secretion in intestinal mucosal cells and enhacnes intestinal wall more resistant to ulceration. Zolimidine exhibits gastroprotective effect in duodenal ulcer research .
    Zolimidine
  • HY-19586
    Albifylline

    A 81-3138; HWA-138

    		 Phosphodiesterase (PDE) Endocrinology
    Albifylline (A 81-3138; HWA-138) is a Xanthine (HY-W017389) derivate. Albifylline reduces the shock-induced leukocyte adhesions to the sinusoidal endothelium in the liver after hemorrhagic shock and improves microvascular blood flow in the liver .
    Albifylline
  • HY-154698
    Homouridine

    		Nucleoside Antimetabolite/Analog Cancer
    Homouridine, is an uridine analogue. Homouridine serves as an intermediate to prepare MMP-2 inhibitor (compund I, IC50=150 μM). Homouridine derivate (compund I) also inhibits TNF-α binding to TNF-αR1 .
    Homouridine
  • HY-142693
    Angiogenesis agent 1

    		HIF/HIF Prolyl-Hydroxylase Metabolic Disease
    Angiogenesis agent 1 (compound C-31) is a salidroside-derivated glycoside analogue. Angiogenesis agent 1 is an activator of the HIF-1α pathway. Angiogenesis agent 1 has the potential for the research of diabetic hind limb ischemia .
    Angiogenesis agent 1
  • HY-W278944
    Antiproliferative agent-15

    		Drug Derivative Cancer
    Antiproliferative agent-15 is an thienopyrimidine derivated anticancer agent. Antiproliferative agent-15 shows antiproliferative activity against human colon (HCT116 and HCT15) and brain (LN-229 and GBM-10) cancer cell lines .
    Antiproliferative agent-15
  • HY-117695
    AQC
    3 Publications Verification

    6-Aminoquinolyl-N-hydroxysccinimidyl carbamate

    		 Fluorescent Dye Others
    AQC (6-Aminoquinolyl-N-hydroxysccinimidyl carbamate) is a reagent used for amino acid or protein sequence analysis by HPLC with fluorescence detection. AQC reacts with primary and secondary amino acids to yield fluorescent derivates, allowing amino acid detection at under-picomolar levels .
    AQC
  • HY-136630
    Felotaxel

    SHR110008

    		 Drug Derivative Others
    Felotaxel (SHR110008) is a derivate of Docetaxel (HY-B0011), with antitumor activity and specific pharmacokinetic properties in rats. Felotaxel is rapidly distributed to normal tissues. The kidney is the major excretion organ, and its plasma protein binding capacity is nearly linearly related to concentration.
    Felotaxel
  • HY-137023
    Sulfo-Cy7 amine

    		Fluorescent Dye Others
    Sulfo-Cy7 amine is a cyanine containing a free amine group, which can be conjugated with a variety of functionalities, including NHS esters, and epoxides. This NIR dye amine can be used to derivate various targets by the reaction with electrophilic groups, and also by enzymatical reactions involving transamination.
    Sulfo-Cy7 amine
  • HY-W471938
    Antiproliferative agent-35

    		Drug Derivative Cancer
    Antiproliferative agent-35 (Compound 4) is an anticancer agent derivated from Esculetin (HY-N0284). Antiproliferative agent-35 inhibits the proliferation of B16 and A549 cells, with IC50s of 13.2 and 9.2 μM resspectively .
    Antiproliferative agent-35
  • HY-157914
    Dibenzyl-14-crown-4

    6,6-Dibenzyl-1,4,8,11-tetraoxacyclotetradecane

    		 Biochemical Assay Reagents Others
    Dibenzyl-14-crown-4 (6,6-Dibenzyl-1,4,8,11-tetraoxacyclotetradecane) is a crown ether derivate, which serves as neutral carrier in PVC ion-selective electrode, improves the Li + selectivity against Na + and K + .
    Dibenzyl-14-crown-4
  • HY-B1794
    Thiethylperazine
    1 Publications Verification

    		 Dopamine Receptor Histamine Receptor Bacterial Amyloid-β Infection Neurological Disease
    Thiethylperazine, a phenothiazine derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist. Thiethylperazine is also a selective ABCC1activator that reduces amyloid-β (Aβ) load in mice. Thiethylperazine has anti-emetic, antipsychotic and antimicrobial effects .
    Thiethylperazine
  • HY-107944
    Chlorphenesin carbamate

    Maolate; U 19646

    		 Others Neurological Disease
    Chlorphenesin carbamate is a centrally acting skeletal muscle relaxant, as well as a derivate of Chlorphenesin (HY-A0133). Chlorphenesin carbamate can be used for the research of pain and discomfort related to skeletal muscle trauma and inflammation . Chlorphenesin carbamate is a selective blocker of polysynaptic pathways at the spinal and supra-spinal levels . Antinociceptive effect .
    Chlorphenesin carbamate
  • HY-172509
    N-Tetradecyl-pSar25

    		Biochemical Assay Reagents Others
    N-Tetradecyl-pSar25 is a polysarcosine (pSar) derivative featuring a tetradecyl head group and a 25-mer polysarcosine tail. Sarcosine is an amino acid derivated that is being developed as an alternative to PEG for in vivo applications due to its biodegradability and highly reduced antigenicity. pSar-lipid derivatives such as this may be applied in the development of lipid nanoparticles.
    N-Tetradecyl-pSar25
  • HY-W007390
    Methyl 2-amino-5-bromobenzoate

    		Bacterial Infection
    Methyl 2-amino-5-bromobenzoate (compound 8/12) can be used for synthesis of 2-benzamidobenzoic acids, which are known FabH inhibitors. The derivates also inhibit PqsD, the pqs quorum sensing (QS) system of Pseudomonas aeruginosa, involving the production of a number of virulence factors and biofilm formation .
    Methyl 2-amino-5-bromobenzoate
  • HY-172288
    N-TETAMINE-pSar45

    		Biochemical Assay Reagents Others
    N-TETAMINE-pSar45 is a polysarcosine (pSar) derivative featuring an N-tetamine head group and a 45-mer polysarcosine tail. Sarcosine is an amino acid derivated that is being developed as an alternative to PEG for in vivo applications due to its biodegradability and highly reduced antigenicity. pSar-lipid derivatives such as this may be applied in the development of lipid nanoparticles.
    N-TETAMINE-pSar45
  • HY-172510
    N-Hexadecyl-pSar25

    		Biochemical Assay Reagents Others
    N-Hexadecyl-pSar25 is a polysarcosine (pSar) derivative featuring a hexadecyl head group and a 25-mer polysarcosine tail. Sarcosine is an amino acid derivated that is being developed as an alternative to PEG for in vivo applications due to its biodegradability and highly reduced antigenicity. pSar-lipid derivatives such as this may be applied in the development of lipid nanoparticles.
    N-Hexadecyl-pSar25
  • HY-136429
    Ethylhydrocupreine

    Optochin

    		 Bacterial Parasite Infection
    Ethylhydrocupreine (Optochin) is a quinine derivate with antimicrobial activity against S. pneumoniae. Ethylhydrocupreine also possesses antimalarial activity against Plasmodium falciparum, with an IC50 of 25.75 nM. Ethylhydrocupreine is a Gallus gallus taste 2 receptors (ggTas2r1, ggTas2r2 and ggTas2r7) agonist .
    Ethylhydrocupreine
  • HY-136429A
    Ethylhydrocupreine hydrochloride

    Optochin hydrochloride

    		 Bacterial Parasite Infection
    Ethylhydrocupreine hydrochloride (Optochin hydrochloride) is a quinine derivate with antimicrobial activity against S. pneumoniae. Ethylhydrocupreine hydrochloride also possesses antimalarial activity against Plasmodium falciparum, with an IC50 of 25.75 nM. Ethylhydrocupreine hydrochloride is a Gallus gallus taste 2 receptors (ggTas2r1, ggTas2r2 and ggTas2r7) agonist .
    Ethylhydrocupreine hydrochloride
  • HY-151340
    Antitubercular agent-32

    		Bacterial Infection
    Antitubercular agent-32 is a derivate of Benzothiazinone (HY-13579A), inhibits M. tuberculosis, and shows improved metabolic stability and enhanced water solubility. Antitubercular agent-32 exerts antitubercular effect by targeting decaprenylphosphoryl-β-D-ribose 2’-oxidase (DprE1, IC50=3.9 μM) .
    Antitubercular agent-32
  • HY-113046S
    5-Methyltetrahydrofolic acid-13C5

    5-Methyl THF-13C5; 5-MTHF-13C,d5

    		 Endogenous Metabolite Metabolic Disease
    5-Methyltetrahydrofolic acid- 13C5 is the 13C-labeled 5-Methyltetrahydrofolic acid. 5-Methyltetrahydrofolic acid (5-Methyl THF) is a biologically active form of folic acid. 5-Methyltetrahydrofolic acid is a methylated derivate of tetrahydrofolate. 5-Methyltetrahydrofolic acid is the predominant natural dietary folate and the principal form of folate in plasma and cerebrospinal fluid[1].
    5-Methyltetrahydrofolic acid-13C5
  • HY-B1794A
    Thiethylperazine dimaleate
    1 Publications Verification

    		 Dopamine Receptor Histamine Receptor Bacterial Amyloid-β Infection Neurological Disease
    Thiethylperazine dimaleate, a phenothiazine derivate, is an orally active and potent dopamine D2-receptor and histamine H1-receptor antagonist. Thiethylperazine dimaleate is also a selective ABCC1activator that reduces amyloid-β (Aβ) load in mice. Thiethylperazine dimaleate has anti-emetic, antipsychotic and antimicrobial effects .
    Thiethylperazine dimaleate
  • HY-151358
    SENP2-IN-1

    		E1/E2/E3 Enzyme Cancer
    SENP2-IN-1 (compound 77) is a selective SENP2 inhibitor. SENP2-IN-1 shows inhibitory activities with IC50s of 1.3, 0.69 and 22.7 μM for SENP1, SENP2 and SENP5, respectively. SENP2-IN-1 can be used for the research of cancer .
    SENP2-IN-1
  • HY-136429AR
    Ethylhydrocupreine (hydrochloride) (Standard)

    		Bacterial Parasite Infection
    Ethylhydrocupreine (hydrochloride) (Standard) is the analytical standard of Ethylhydrocupreine (hydrochloride). This product is intended for research and analytical applications. Ethylhydrocupreine hydrochloride (Optochin hydrochloride) is a quinine derivate with antimicrobial activity against S. pneumoniae. Ethylhydrocupreine hydrochloride also possesses antimalarial activity against Plasmodium falciparum, with an IC50 of 25.75 nM. Ethylhydrocupreine hydrochloride is a Gallus gallus taste 2 receptors (ggTas2r1, ggTas2r2 and ggTas2r7) agonist .
    Ethylhydrocupreine (hydrochloride) (Standard)

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