Search Result
Results for "
psychoactivity
" in MedChemExpress (MCE) Product Catalog:
1
Biochemical Assay Reagents
3
Isotope-Labeled Compounds
Cat. No. |
Product Name |
Target |
Research Areas |
Chemical Structure |
-
- HY-116795
-
|
Others
|
Neurological Disease
|
5-Methoxy-α-ethyltryptamine is a tryptamine psychoactive substance, which has nerve stimulated effect .
|
-
-
- HY-137994
-
|
Others
|
Neurological Disease
|
Deschloroetizolam is a designer Benzodiazepine. Deschloroetizolam is a psychoactive substance, with physical and cognitive effects .
|
-
-
- HY-W783639
-
-
-
- HY-129850
-
-
-
- HY-168014
-
-
-
- HY-169465
-
-
-
- HY-W753724
-
-
-
- HY-169447
-
-
-
- HY-117526
-
-
-
- HY-59059
-
|
Monoamine Oxidase
|
Neurological Disease
|
5-(2-Aminopropyl)indole is an orally active psychoactive substance, that shows inhibitory activity against monoamine oxidase (MAO) and long-lasting stimulatory properties .
|
-
-
- HY-121870A
-
Larocaine hydrochloride
|
Dopamine Receptor
|
Neurological Disease
|
Dimethocaine (Larocaine) hydrochloride is distributed and consumed as "new psychoactive substance" (NPS) without any safety testing
|
-
-
- HY-137979
-
|
Others
|
Neurological Disease
|
Flunitrazolam is an orally active designer Benzodiazepine. Flunitrazolam is biologically toxic, class in psychoactive substances .
|
-
-
- HY-135154
-
|
GABA Receptor
|
Neurological Disease
|
epi-Aszonalenin A is a benzodiazepine fungal metabolite originally isolated from Aspergillus novofumigatus. epi-Aszonalenin A can be used as a psychoactive agent .
|
-
-
- HY-A0171
-
Ba-30803 free base
|
5-HT Receptor
|
Neurological Disease
|
Benzoctamine is an orally active and potent psychoactive agent which possesses tranquillizing properties. Benzoctamine increases the turnover rate of catecholamines. Benzoctamine enhances the [3H]noradrenaline uptake in the rat heart. Benzoctamine also accelerated the disappearance of intracisternally injected [3H]noradrenaline .
|
-
-
- HY-105927
-
-
-
- HY-W718081
-
-
-
- HY-B0188
-
-
-
- HY-139237
-
|
Drug Derivative
|
Neurological Disease
|
PCEEA hydrochloride is a synthetic agent which is structurally related to the psychoactive compounds Eticyclidine, Ketamine, and Phencyclidine.
|
-
-
- HY-158554
-
2-Eec hydrochloride
|
Biochemical Assay Reagents
|
Others
|
2-Ethylethcathinone hydrochloride (2-Eec hydrochloride) is a substituted cathinone (compounds with potential for abuse). 2-Ethylethcathinone hydrochloride is a stereoisomer of 2-fluoroethcathinone .
|
-
-
- HY-W098756
-
-
-
- HY-B0188A
-
-
-
- HY-W721259
-
|
Drug Isomer
|
Others
|
2-Bromoamphetamine hydrochloride is an isomer of 4-Bromoamphetamine. 4-Bromoamphetamine is a psychoactive substance .
|
-
-
- HY-172071
-
PAL-1046 hydrochloride
|
5-HT Receptor
|
Neurological Disease
|
Methamnetamine (PAL-1046) hydrochloride is an amphetamine-based psychoactive substance. Methamnetamine hydrochloride causes excessive release of serotonin .
|
-
-
- HY-W028389
-
|
GABA Receptor
|
Neurological Disease
|
Pyrazolam, a Benzodiazepines psychoactive substance, is a central nervous system depressant. Pyrazolam can cause psychomotor impairment .
|
-
-
- HY-N0700
-
α-Asarone; trans-Asarone
|
GABA Receptor
|
Neurological Disease
|
alpha-Asarone (α-Asarone) is one of the main psychoactive compounds, and possesses an antidepressant-like activity in mice.
|
-
-
- HY-W775306
-
-
-
- HY-W008150
-
-
-
- HY-W014971
-
|
Biochemical Assay Reagents
|
Others
|
Tryptamine hydrochloride belongs to the class of indole alkaloids and is a derivative of the amino acid tryptophan. Tryptamine hydrochloride is psychoactive and acts as a neurotransmitter in the body, affecting mood, perception and cognition. In its hydrochloride form, Tryptamine hydrochloride hydrochloride, it is commonly used as a research chemical and as a starting material for the synthesis of other organic compounds. It can also occur naturally in certain plants and animals, including fungi and mammals. Due to the psychoactive properties of Tryptamine hydrochloride and its derivatives, its use and possession are controlled substances in many countries.
|
-
-
- HY-B0188AS
-
Org GB 94-d3
|
Histamine Receptor
|
Neurological Disease
Endocrinology
|
Mianserin-d3 (hydrochloride) is the deuterium labeled Mianserin hydrochloride. Mianserin hydrochloride (Org GB 94) is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
|
-
-
- HY-137429
-
Acidum valiloxibicum; XWL-008
|
GABA Receptor
|
Neurological Disease
|
Valiloxibic acid is a proagent of γ-Hydroxybutyric acid (GHB).GHB is a naturally occurring neurotransmitter and a psychoactive agent, it acts on the GHB receptor and is a weak agonist at the GABAB receptor .
|
-
-
- HY-169448
-
EPT
|
5-HT Receptor
|
Others
|
Ethylpropyltryptamine (EPT) is a novel orally active psychoactive substance. Ethylpropyltryptamine (EPT) is predicted to be a partial agonist of the 5-HT2A receptor .
|
-
-
- HY-169442
-
|
Biochemical Assay Reagents
|
Neurological Disease
|
Methylmethaqualone is a quinazolinone psychoactive substance that can be used as an analytical reference standard for quinazolinone compounds. Methylmethaqualone has acute neurotoxicity and can cause psychomotor stimulation .
|
-
-
- HY-U00241
-
RGH 3331; Uxepam
|
GABA Receptor
|
Neurological Disease
|
Carburazepam is a agent which derives from benzodiazepine. Benzodiazepines (BZD, BZs) are a class of psychoactive agents whose core chemical structure is the fusion of a benzene ring and a diazepine ring.
|
-
-
- HY-122303
-
|
5-HT Receptor
|
Neurological Disease
|
4-hydroxy DiPT hydrochloride is an 5-HT2A agonist that induces the head-twitch response (HTR) in mice, indicating psychoactivity .
|
-
-
- HY-W721302
-
|
Monoamine Oxidase
|
Neurological Disease
|
2-APB is an analog of 6-APB, a benzofuran derivative and a psychoactive substance. Certain benzofuran derivatives have monoamine oxidase-A inhibitory activity .
|
-
-
- HY-B0188S
-
-
-
- HY-172030
-
-
-
- HY-A0171A
-
Ba-30803
|
5-HT Receptor
|
Neurological Disease
|
Benzoctamine hydrochloride (Ba-30803) is a psychoactive agent with anti-anxiety effect. Benzoctamine hydrochloride blocks the central postsynaptic serotonin receptors and decreases 5-HT turnover in the brain .
|
-
-
- HY-B0188AR
-
|
Histamine Receptor
|
Neurological Disease
Endocrinology
|
Mianserin (hydrochloride) (Standard) is the analytical standard of Mianserin (hydrochloride). This product is intended for research and analytical applications. Mianserin hydrochloride (Org GB 94) is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
|
-
-
- HY-W1023070
-
|
5-HT Receptor
|
Neurological Disease
|
4-fluoro MBZP is a new psychoactive substance that belongs to the phenylpiperazine class of compounds and can be used to study the 5-HT2 receptors in the central nervous system .
|
-
-
- HY-N0700R
-
|
GABA Receptor
|
Neurological Disease
|
alpha-Asarone (Standard) is the analytical standard of alpha-Asarone. This product is intended for research and analytical applications. alpha-Asarone (α-Asarone) is one of the main psychoactive compounds, and possesses an antidepressant-like activity in mice.
|
-
-
- HY-B0489A
-
-
-
- HY-N2364
-
-
-
- HY-118796
-
4-HO-MET; 4-Hydroxy-N-methyl-N-ethyltryptamine
|
5-HT Receptor
|
Neurological Disease
|
4-Hydroxy MET (4-HO-MET) is a psychoactive tryptamine (NPS), a structural variant of the endogenous neurotransmitter serotonin. 4-Hydroxy MET has hallucinogenic effects, affecting mood, movement, and cognitive function .
|
-
-
- HY-120243
-
|
iGluR
|
Neurological Disease
|
L-Ibotenic acid is a psychoactive compound found in Amanita muscaria and related mushroom species. L-Ibotenic acid is a conformationally restricted analog of the neurotransmitter glutamate, which may be activated by different conformations of L-glutamate and is a non-selective glutamate receptor agonist .
|
-
-
- HY-170310
-
|
Opioid Receptor
|
Neurological Disease
|
AP-238 is a a new synthetic opioid (NSO), and acts as an agonist for μ-opioid receptor (MOR) with an EC50 of 248 nM. AP-238 exhibits analgesic activity .
|
-
-
- HY-103092
-
|
5-HT Receptor
|
Neurological Disease
|
CP-135807 is an orally active and selective 5-HT1D agonist (IC50=3.1 nM), bovine). CP-135807 mediates central psychoactivity and can be used in antidepressant research .
|
-
-
- HY-B0489
-
methyl 1,2,5,6-tetrahydro-1-methyl-3-pyridinecarboxylate hydrobromide
|
mAChR
nAChR
|
Infection
Neurological Disease
Metabolic Disease
Inflammation/Immunology
Cancer
|
Arecoline hydrobromide, a naturally occurring psychoactive alkaloid, is a partial agonist of nicotinic and muscarinic acetylcholine receptor. Arecoline hydrobromide exhibits stimulation, alertness, anxiolysis and anti-parasitic effects. Arecoline hydrobromide also can induce oxidative stress .
|
-
-
- HY-W783639S
-
-
-
- HY-169466
-
|
Drug Derivative
|
Neurological Disease
|
5-Methoxy-N,N-dimethyltryptamine Nb-oxide is an indole alkaloid. 5-Methoxy-N,N-dimethyltryptamine Nb-oxide is the N-oxide form of 5-Methoxy-N,N-dimethyltryptamine (5-MeO-DMT), which is a known psychoactive substance .
|
-
- HY-135222
-
5-Methoxy-6-methyl-2-aminoindan hydrochloride
|
5-HT Receptor
|
Neurological Disease
|
MMAI (5-Methoxy-6-methyl-2-aminoindan) hydrochloride is a selective serotonin releaser that does not produce psychoactive or hallucinogenic effects in the context of drug discrimination in rats. MMAI hydrochloride induces a behavioral syndrome in rats, including hypokinesia with freezing, spinning, Straub tail, flat posture, and reduced sleep time .
|
-
- HY-W742532
-
N-Ethyl-nor-LSD
|
5-HT Receptor
Dopamine Receptor
|
Neurological Disease
|
ETH-LAD (N-Ethyl-nor-LSD) is an activator for 5-HT2A receptor with Ki of 5.1 nM. ETH-LAD exhibits affinity for dopamine receptor D1 and dopamine receptor D2 with Ki of 22.1 nM and 4.4 nM. ETH-LAD acts as psychoactive substance in rat model .
|
-
- HY-169785
-
7-TMT
|
5-HT Receptor
|
Neurological Disease
|
7-Methyl DMT (7-TMT) is a 5-HT2 receptor agonist. Structurally, 7-Methyl DMT is a tryptamine derivative. It can be used as an analytical reference standard for the psychoactive substance DOM. 7-Methyl DMT is also used in research in the field of neurological diseases .
|
-
- HY-B0489R
-
|
mAChR
nAChR
|
Infection
Neurological Disease
Metabolic Disease
Inflammation/Immunology
Cancer
|
Arecoline (hydrobromide) (Standard) is the analytical standard of Arecoline (hydrobromide). This product is intended for research and analytical applications. Arecoline hydrobromide, a naturally occurring psychoactive alkaloid, is a partial agonist of nicotinic and muscarinic acetylcholine receptor. Arecoline hydrobromide exhibits stimulation, alertness, anxiolysis and anti-parasitic effects. Arecoline hydrobromide also can induce oxidative stress .
|
-
- HY-W775346
-
Δ8-THC acetate; Delta8-tetrahydrocannabinol
|
Cannabinoid Receptor
|
Neurological Disease
Inflammation/Immunology
|
Delta8-THC acetate (Delta8-tetrahydrocannabinol) is a psychoactive phytocannabinoid, that binds to cannabinoid receptor 1 (CB1 receptor), and exhibits anti-nausea, appetite-stimulating, and anti-inflammatory activities. Delta8-THC acetate exhibits probably neuroprotective efficacy and can be used in anti-anxiety and antidepressant research .
|
-
- HY-W743888
-
6-Allyl-6-nor-LSD
|
5-HT Receptor
Dopamine Receptor
|
Neurological Disease
|
AL-LAD (6-Allyl-6-nor-LSD) is an activator for 5-HT2A receptor with Ki of 3.4-8.1 nM. AL-LAD exhibits affinity for dopamine receptor D1 and dopamine receptor D2 with absolute affinitiesK0.5 of 189 nM and 12.3 nM. AL-LAD acts as psychoactive substance in mouse model .
|
-
- HY-B1033
-
|
5-HT Receptor
Dopamine Receptor
Sodium Channel
|
Neurological Disease
|
Metergoline is a serotonin (5-HT) receptor and dopamine receptors antagonist, with pKis of 8.64, 8.75 and 8.75 for 5-HT2A, 5-HT2B and 5-HT2C, respectively. Metergoline is a high-affinity ligand for the h5-HT7 receptor, with a Ki of 16 nM. Metergoline is also a reversible neural Na + channels inhibitor. Metergoline is commonly used for the research of seasonal affective disorder, prolactin hormone regulation .
|
-
- HY-108295
-
CXB-722
|
GABA Receptor
|
Neurological Disease
|
Pivagabine (CXB 722) is a hydrophobic 4-aminobutyric acid derivative with neuromodulatory activity. Pivagabine penetrates the blood-brain barrier in rats. Pivagabine antagonizes the effects of foot shock on both GABAA receptor function and corticotropin-releasing factor (CRF) concentrations in rat brain .
|
-
- HY-117087
-
|
Phosphatase
|
Cancer
|
K103 is an inhibitor discovered from the screen that is an analog of the serotonin antagonist benzazocine. K103 exhibited inhibition of SHIP homologues, labelling it a pan-SHIP1/2 inhibitor, but the molecule had no effect on another 5' inositol phosphatase, OCRL. In line with the "two PIPs hypothesis", the molecule exhibited significant anti-tumour effects against a variety of cell lines, particularly breast cancer cells. Additional studies with K103 revealed that inhibition of SHIP1/2 in multiple myeloma cells resulted in G2/M cell cycle arrest followed by extensive apoptosis via activation of the caspase cascade. K103 fits the commonly used small molecule agent property profile, but while this work was being conducted, it was discovered that K103 caused psychoactive effects in mice, which limited the utility of the molecule in vivo. Therefore, certain synthetic studies were conducted on this tryptamine to identify the features that needed to be present in the molecule to maintain pan-SHIP1/2 inhibition in order to design an inhibitor with favourable pharmacodynamic properties and an improved side effect profile.
|
-
Cat. No. |
Product Name |
Type |
-
- HY-W014971
-
|
Biochemical Assay Reagents
|
Tryptamine hydrochloride belongs to the class of indole alkaloids and is a derivative of the amino acid tryptophan. Tryptamine hydrochloride is psychoactive and acts as a neurotransmitter in the body, affecting mood, perception and cognition. In its hydrochloride form, Tryptamine hydrochloride hydrochloride, it is commonly used as a research chemical and as a starting material for the synthesis of other organic compounds. It can also occur naturally in certain plants and animals, including fungi and mammals. Due to the psychoactive properties of Tryptamine hydrochloride and its derivatives, its use and possession are controlled substances in many countries.
|
Cat. No. |
Product Name |
Category |
Target |
Chemical Structure |
Cat. No. |
Product Name |
Chemical Structure |
-
- HY-B0188AS
-
|
Mianserin-d3 (hydrochloride) is the deuterium labeled Mianserin hydrochloride. Mianserin hydrochloride (Org GB 94) is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
|
-
-
- HY-B0188S
-
|
Mianserin-d3 is the deuterium labeled Mianserin (HY-B0188). Mianserin? is a Histamine 1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant .
|
-
-
- HY-W783639S
-
|
Bzo-poxizid-d9 (5C-MDA-19-d9, Petyl MDA-19-d9) is deuterium labeled Bzo-poxizid. Bzo-poxizid is a synthetic cannabinoid that is a psychoactive substance .
|
-
Your information is safe with us. * Required Fields.
Inquiry Information
- Product Name:
- Cat. No.:
- Quantity:
- MCE Japan Authorized Agent: