2. Vitamin D Related/Nuclear Receptor
  3. Estrogen Receptor/ERR
  4. Pipendoxifene hydrochloride

Pipendoxifene hydrochloride is a selective estrogen receptor modulator (SERM) that can be used for the research of breast cancer.

For research use only. We do not sell to patients.

Pipendoxifene hydrochloride Chemical Structure

Pipendoxifene hydrochloride Chemical Structure

CAS No. : 245124-69-0

Size Price Stock Quantity
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO
ready for reconstitution
 USD 154 In-stock
Solution
10 mM * 1 mL in DMSO USD 154 In-stock
Solid
5 mg USD 140 In-stock
10 mg USD 230 In-stock
25 mg USD 480 In-stock
50 mg USD 800 In-stock
100 mg USD 1350 In-stock
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of Pipendoxifene hydrochloride:

Pipendoxifene hydrochloride Related Antibodies

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Estrogen receptor ERα ERβ ERRα ERRβ ERRγ

  • Biological Activity

  • Purity & Documentation

  • References

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Description

Pipendoxifene hydrochloride is a selective estrogen receptor modulator (SERM) that can be used for the research of breast cancer[1].

IC50 & Target

Estrogen receptor[1]
In Vitro

Pipendoxifene is a new 2-phenyl indole selective estrogen receptor modulators (SERM) that exhibits an excellent preclinical pharmacological profile and is selected for further development as a treatment for metastatic breast cancer[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Pipendoxifene hydrochloride Related Antibodies
Molecular Weight

493.04

Formula

C29H33ClN2O3
CAS No.
Appearance

Solid

Color

White to yellow

SMILES

OC1=CC2=C(N(CC3=CC=C(OCCN4CCCCC4)C=C3)C(C5=CC=C(O)C=C5)=C2C)C=C1.Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (202.82 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.0282 mL 10.1412 mL 20.2823 mL
5 mM 0.4056 mL 2.0282 mL 4.0565 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Purity: 99.83%

COA (252 KB) LCMS (94 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.0282 mL 10.1412 mL 20.2823 mL 50.7058 mL
5 mM 0.4056 mL 2.0282 mL 4.0565 mL 10.1412 mL
10 mM 0.2028 mL 1.0141 mL 2.0282 mL 5.0706 mL
15 mM 0.1352 mL 0.6761 mL 1.3522 mL 3.3804 mL
20 mM 0.1014 mL 0.5071 mL 1.0141 mL 2.5353 mL
25 mM 0.0811 mL 0.4056 mL 0.8113 mL 2.0282 mL
30 mM 0.0676 mL 0.3380 mL 0.6761 mL 1.6902 mL
40 mM 0.0507 mL 0.2535 mL 0.5071 mL 1.2676 mL
50 mM 0.0406 mL 0.2028 mL 0.4056 mL 1.0141 mL
60 mM 0.0338 mL 0.1690 mL 0.3380 mL 0.8451 mL
80 mM 0.0254 mL 0.1268 mL 0.2535 mL 0.6338 mL
100 mM 0.0203 mL 0.1014 mL 0.2028 mL 0.5071 mL
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Pipendoxifene hydrochloride Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Pipendoxifene245124-69-0Estrogen Receptor/ERRInhibitorinhibitorinhibit

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