Pipendoxifene hydrochloride

Name: Pipendoxifene hydrochloride
Brand: MedChemExpress
SKU: HY-13724B
Rating: 4.5 (1 reviews)

Cat. No.: HY-13724B Purity: 99.83%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

Pipendoxifene hydrochloride is a selective estrogen receptor modulator (SERM) that can be used for the research of breast cancer.

For research use only. We do not sell to patients.

Pipendoxifene hydrochloride Chemical Structure

CAS No. : 245124-69-0

Size	Price	Stock	Quantity
Solid + Solvent (Highly Recommended)
10 mM * 1 mL in DMSO ready for reconstitution	USD 154	In-stock	Estimated Time of Arrival: December 31
Solution
10 mM * 1 mL in DMSO	USD 154	In-stock	Estimated Time of Arrival: December 31
Solid
5 mg	USD 140	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 230	In-stock	Estimated Time of Arrival: December 31
25 mg	USD 480	In-stock	Estimated Time of Arrival: December 31
50 mg	USD 800	In-stock	Estimated Time of Arrival: December 31
100 mg	USD 1350	In-stock	Estimated Time of Arrival: December 31
200 mg		Get quote
500 mg		Get quote

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Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of Pipendoxifene hydrochloride:

Pipendoxifene Get quote

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Biological Activity
Purity & Documentation
References
Customer Review

Description

Pipendoxifene hydrochloride is a selective estrogen receptor modulator (SERM) that can be used for the research of breast cancer^[1].

IC₅₀ & Target

Estrogen receptor^[1]

In Vitro

Pipendoxifene is a new 2-phenyl indole selective estrogen receptor modulators (SERM) that exhibits an excellent preclinical pharmacological profile and is selected for further development as a treatment for metastatic breast cancer^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

493.04

Formula

C₂₉H₃₃ClN₂O₃

CAS No.

245124-69-0

Appearance

Solid

Color

White to yellow

SMILES

OC1=CC2=C(N(CC3=CC=C(OCCN4CCCCC4)C=C3)C(C5=CC=C(O)C=C5)=C2C)C=C1.Cl

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility

In Vitro:

DMSO : 100 mg/mL (202.82 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.0282 mL	10.1412 mL	20.2823 mL
5 mM	0.4056 mL	2.0282 mL	4.0565 mL
10 mM	0.2028 mL	1.0141 mL	2.0282 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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Volume _(start)

Concentration _(final)

Volume _(final)

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: 99.83%

Select Batch:

Data Sheet (272 KB) SDS (393 KB)

COA (252 KB) LCMS (94 KB)

Handling Instructions (2659 KB)

References

[1]. Shelly W, et al. Selective estrogen receptor modulators: an update on recent clinical findings. Obstet Gynecol Surv. 2008 Mar;63(3):163-81. [Content Brief]

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	2.0282 mL	10.1412 mL	20.2823 mL	50.7058 mL
	5 mM	0.4056 mL	2.0282 mL	4.0565 mL	10.1412 mL
	10 mM	0.2028 mL	1.0141 mL	2.0282 mL	5.0706 mL
	15 mM	0.1352 mL	0.6761 mL	1.3522 mL	3.3804 mL
	20 mM	0.1014 mL	0.5071 mL	1.0141 mL	2.5353 mL
	25 mM	0.0811 mL	0.4056 mL	0.8113 mL	2.0282 mL
	30 mM	0.0676 mL	0.3380 mL	0.6761 mL	1.6902 mL
	40 mM	0.0507 mL	0.2535 mL	0.5071 mL	1.2676 mL
	50 mM	0.0406 mL	0.2028 mL	0.4056 mL	1.0141 mL
	60 mM	0.0338 mL	0.1690 mL	0.3380 mL	0.8451 mL
	80 mM	0.0254 mL	0.1268 mL	0.2535 mL	0.6338 mL
	100 mM	0.0203 mL	0.1014 mL	0.2028 mL	0.5071 mL