FBPase-1 inhibitor-1

Cat. No.: HY-136717 Purity: 99.10%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

FBPase-1 inhibitor-1 (compound 1) is a allosteric inhibitor of fructose-1,6-bisphosphatase (FBPase-1).

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FBPase-1 inhibitor-1 Chemical Structure

CAS No. : 883973-99-7

Size	Price	Stock	Quantity
Free Sample (0.1 - 0.5 mg)		Apply Now
5 mg	USD 66	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 106	In-stock	Estimated Time of Arrival: December 31
25 mg	USD 211	In-stock	Estimated Time of Arrival: December 31
50 mg	USD 338	In-stock	Estimated Time of Arrival: December 31
100 mg	USD 540	In-stock	Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

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Purity & Documentation
References
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Description

FBPase-1 inhibitor-1 (compound 1) is a allosteric inhibitor of fructose-1,6-bisphosphatase (FBPase-1)^[1].

Molecular Weight

377.63

Formula

C₁₃H₇Cl₃N₂O₃S

CAS No.

883973-99-7

Appearance

Solid

Color

White to off-white

SMILES

O=S(C1=CC(Cl)=CC=C1Cl)(NC2=NC3=CC(Cl)=CC=C3O2)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Solvent & Solubility

In Vitro:

DMSO : 125 mg/mL (331.01 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.6481 mL	13.2405 mL	26.4809 mL
5 mM	0.5296 mL	2.6481 mL	5.2962 mL
10 mM	0.2648 mL	1.3240 mL	2.6481 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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Concentration _(final)

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Working solution concentration: mg/mL

Purity & Documentation

Purity: 99.10%

Select Batch:

Data Sheet (269 KB) SDS (393 KB)

COA (249 KB) LCMS (94 KB)

Handling Instructions (2659 KB)

References

[1]. Thomas W von Geldern, et al. Benzoxazole benzenesulfonamides are novel allosteric inhibitors of fructose-1,6-bisphosphatase with a distinct binding mode. Bioorg Med Chem Lett. 2006 Apr 1;16(7):1811-5. [Content Brief]

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	2.6481 mL	13.2405 mL	26.4809 mL	66.2024 mL
	5 mM	0.5296 mL	2.6481 mL	5.2962 mL	13.2405 mL
	10 mM	0.2648 mL	1.3240 mL	2.6481 mL	6.6202 mL
	15 mM	0.1765 mL	0.8827 mL	1.7654 mL	4.4135 mL
	20 mM	0.1324 mL	0.6620 mL	1.3240 mL	3.3101 mL
	25 mM	0.1059 mL	0.5296 mL	1.0592 mL	2.6481 mL
	30 mM	0.0883 mL	0.4413 mL	0.8827 mL	2.2067 mL
	40 mM	0.0662 mL	0.3310 mL	0.6620 mL	1.6551 mL
	50 mM	0.0530 mL	0.2648 mL	0.5296 mL	1.3240 mL
	60 mM	0.0441 mL	0.2207 mL	0.4413 mL	1.1034 mL
	80 mM	0.0331 mL	0.1655 mL	0.3310 mL	0.8275 mL
	100 mM	0.0265 mL	0.1324 mL	0.2648 mL	0.6620 mL