2. Protein Tyrosine Kinase/RTK
  3. Src
  4. Lck-IN-1

Lck-IN-1 is a potent lymphocyte protein tyrosine kinase (Lck) inhibitor extracted from patent WO2007013673A1, example 48.

For research use only. We do not sell to patients.

Lck-IN-1 Chemical Structure

Lck-IN-1 Chemical Structure

CAS No. : 923596-52-5

Size Price Stock Quantity
5 mg In-stock
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50 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Lck Fyn Blk Hck Lyn Yes

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Description

Lck-IN-1 is a potent lymphocyte protein tyrosine kinase (Lck) inhibitor extracted from patent WO2007013673A1, example 48[1].

Molecular Weight

253.30

Formula

C14H15N5
CAS No.
Appearance

Solid

Color

Light yellow to yellow

SMILES

CCCNC1=NN2C(C=C1)=NC=C2C3=CC=NC=C3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

-20°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (394.79 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 3.9479 mL 19.7394 mL 39.4789 mL
5 mM 0.7896 mL 3.9479 mL 7.8958 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

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Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
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Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (protect from light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 3.9479 mL 19.7394 mL 39.4789 mL 98.6972 mL
5 mM 0.7896 mL 3.9479 mL 7.8958 mL 19.7394 mL
10 mM 0.3948 mL 1.9739 mL 3.9479 mL 9.8697 mL
15 mM 0.2632 mL 1.3160 mL 2.6319 mL 6.5798 mL
20 mM 0.1974 mL 0.9870 mL 1.9739 mL 4.9349 mL
25 mM 0.1579 mL 0.7896 mL 1.5792 mL 3.9479 mL
30 mM 0.1316 mL 0.6580 mL 1.3160 mL 3.2899 mL
40 mM 0.0987 mL 0.4935 mL 0.9870 mL 2.4674 mL
50 mM 0.0790 mL 0.3948 mL 0.7896 mL 1.9739 mL
60 mM 0.0658 mL 0.3290 mL 0.6580 mL 1.6450 mL
80 mM 0.0493 mL 0.2467 mL 0.4935 mL 1.2337 mL
100 mM 0.0395 mL 0.1974 mL 0.3948 mL 0.9870 mL
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Lck-IN-1 Related Classifications

Keywords:

Lck-IN-1923596-52-5SrcInhibitorinhibitorinhibit

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