MK-761 free base

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MK-761 free base is a potent and orally active β2-adrenergic blocker. MK-761 free base shows antihypertensive and positive inotropic effects. MK-761 free base shows vasodilating properties.

For research use only. We do not sell to patients.

MK-761 free base Chemical Structure

CAS No. : 65321-41-7

Size	Price	Stock	Quantity
5 mg	USD 359	Get quote 2 - 4 weeks 2 - 4 weeks 1 - 3 weeks	Estimated Time of Arrival: December 31
10 mg	USD 597	Get quote 2 - 4 weeks 2 - 4 weeks 1 - 3 weeks	Estimated Time of Arrival: December 31
25 mg	USD 1225	Get quote 2 - 4 weeks 2 - 4 weeks 1 - 3 weeks	Estimated Time of Arrival: December 31
50 mg		Get quote
100 mg		Get quote

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α adrenergic receptor β adrenergic receptor

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Description

MK-761 free base is a potent and orally active β2-adrenergic blocker. MK-761 free base shows antihypertensive and positive inotropic effects. MK-761 free base shows vasodilating properties^[1].

IC₅₀ & Target^[1]

Beta-2 adrenergic receptor

Molecular Weight

249.31

Formula

C₁₃H₁₉N₃O₂

CAS No.

65321-41-7

SMILES

N#CC1=CC=CN=C1OC[C@H](CNC(C)(C)C)O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Handling Instructions (2659 KB)

References

[1]. Scriabine A, et al. Antihypertensive and cardiac effects of two novel beta-adrenoceptor blocking drugs. Experientia. 1979 Dec 15;35(12):1634-7. [Content Brief]

[2]. C.S. Sweet, et al. Peripheral Vasodilator and β-Adrenoceptor Blocking Properties of Several β-Adrenoceptor Antagonists. Clinical and Experimental Hypertension. 2009, 449-471.

[3]. Sweet CS, et al. Beta adrenoceptor blocking properties of MK-761. J Pharmacol Exp Ther. 1979 Oct;211(1):195-9. [Content Brief]

MK-761 free base Related Classifications

Cardiovascular Disease

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)	×	Volume _(start)	=	Concentration _(final)	×	Volume _(final)
	×		=		×
C1		V1		C2		V2

Help & FAQs

Do most proteins show cross-species activity?
Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MK-76165321-41-7MK761MK 761Adrenergic ReceptorBeta Receptororally activeantihypertensivevasodilating propertiesInhibitorinhibitorinhibit

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