1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
  3. P2X Receptor
  4. P2X Receptor Inhibitors

P2X Receptor Inhibitors

P2X1 Receptor

P2X2 Receptor

P2X3 Receptor

P2X4 Receptor

P2X7 Receptor

Your Search Returned No Results.

Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

P2X Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name P2X1 Receptor P2X2 Receptor P2X3 Receptor P2X4 Receptor P2X7 Receptor Purity
BzATP triethylammonium salt
p2x1 Receptor
 
P2X3 Receptor
P2X4 Receptor
P2X7 Receptor
A-740003        
P2X7 Receptor
99.59%
Sodium metatungstate        
P2X7 Receptor
KN-62        
P2X7 Receptor
99.45%
NF449 octasodium
p2x1 Receptor
        ≥99.0%
HEI3090        
P2X7 Receptor
NF449
p2x1 Receptor
       
A 438079 hydrochloride        
P2X7 Receptor
99.92%
Aurintricarboxylic acid
p2x1 Receptor, IC50: 8.6 nM
 
P2X3 Receptor, IC50: 72.9 nM
   
Gefapixant    
P2X3 Receptor
    99.32%
A 438079        
P2X7 Receptor
99.88%
5-BDBD      
P2X4 Receptor
  99.94%
α,β-Methylene-ATP trisodium
p2x1 Receptor
 
P2X3 Receptor
 
P2X7 Receptor
99.75%
JNJ-47965567        
P2X7 Receptor
99.79%
PPADS tetrasodium
p2x1 Receptor
       
BAY-1797      
P2X4 Receptor
  99.42%
AZD9056 hydrochloride        
P2X7 Receptor
98.82%
AZ10606120 dihydrochloride        
P2X7 Receptor
99.38%
A-317491    
P2X3 Receptor
    98.77%
PSB-12062      
P2X4 Receptor
  98.70%
NF023 hexasodium
p2x1 Receptor
        ≥99.0%
A-804598        
P2X7 Receptor
98.55%
PPNDS tetrasodium
p2x1 Receptor
       
P2X3 antagonist 34    
P2X3 Receptor
    99.71%
BX430      
P2X4 Receptor
  99.83%
GSK-1482160        
P2X7 Receptor
98.20%
Minodronic acid  
P2X2 Receptor
P2X3 Receptor
    ≥98.0%
Oxatomide        
P2X7 Receptor
99.56%
Opiranserin hydrochloride    
P2X3 Receptor
    99.44%
A-317491 sodium salt hydrate    
P2X3 Receptor
    99.88%
Bullatine A        
P2X7 Receptor
≥98.0%
NF279
p2x1 Receptor
        ≥98.0%
Lu AF27139        
P2X7 Receptor
99.71%
Oxidized ATP trisodium salt        
P2X7 Receptor
≥98.0%
Gardenoside    
P2X3 Receptor
 
P2X7 Receptor
99.55%
GW791343 dihydrochloride        
P2X7 Receptor, pIC50: 6.9-7.2
98.03%
EVT-401        
P2X7 Receptor
99.89%
RO-3  
P2X2 Receptor
P2X3 Receptor
   
Gefapixant citrate    
P2X3 Receptor
   
Blue FPG-A trisodium
p2x1 Receptor, IC50: 35.5 μM
       
P2X3 antagonist 38    
P2X3 Receptor, IC50: 0.132 μM
   
Minodronic acid-d4  
P2X2 Receptor
P2X3 Receptor
   
(S)-JNJ-54166060        
P2X7 Receptor
P2X4 antagonist-2      
P2X4 Receptor, IC50: 24 nM
 
P2X4 antagonist-1      
P2X4 Receptor, IC50: 15 nM
 
P2X7 receptor antagonist-3        
hP2X7R, IC50: 4.2 nM
rP2X7R, IC50: 6.8 nM
Opiranserin    
P2X3 Receptor
   
PPADS
p2x1 Receptor, IC50: 68 nM
P2X2 Receptor, IC50: 214 nM
     
α,β-Methylene-ATP dilithium
p2x1 Receptor
 
P2X3 Receptor
 
P2X7 Receptor
GW791343 trihydrochloride        
P2X7 Receptor, pIC50: 6.9-7.2