2. GPCR/G Protein Neuronal Signaling Metabolic Enzyme/Protease
  3. 5-HT Receptor Drug Metabolite
  4. Ketanserinol

Ketanserinol  (Synonyms: R 46742)

Cat. No.: HY-121208 Purity: 98.05%
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Ketanserinol (R 46742) is a metabolite of Ketanserin (HY-10562). Ketanserinol is a competitive antagonist of the effects of 5-HT (HY-B1473A) in both arteries. The KB values are 6.5 for large coronary arteries and 6.4 for pulmonary arteries.

For research use only. We do not sell to patients.

Ketanserinol Chemical Structure

Ketanserinol Chemical Structure

CAS No. : 76330-73-9

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Based on 1 publication(s) in Google Scholar

Ketanserinol Related Antibodies

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Description

Ketanserinol (R 46742) is a metabolite of Ketanserin (HY-10562). Ketanserinol is a competitive antagonist of the effects of 5-HT (HY-B1473A) in both arteries. The KB values are 6.5 for large coronary arteries and 6.4 for pulmonary arteries[1].

Molecular Weight

397.44

Formula

C22H24FN3O3
CAS No.
Appearance

Solid

SMILES

O=C(NC1=C(C2=O)C=CC=C1)N2CCN3CCC(CC3)C(O)C4=CC=C(C=C4)F
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

4°C, protect from light

*In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)

Purity & Documentation

Purity: 98.05%

COA (246 KB) HNMR (222 KB) LCMS (140 KB)

Handling Instructions (2659 KB)
References
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Ketanserinol Related Classifications

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Ketanserinol76330-73-9R 46742R46742R-467425-HT ReceptorDrug MetaboliteSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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