2. GPCR/G Protein Neuronal Signaling
  3. Somatostatin Receptor
  4. NODAGA-LM3

NODAGA-LM3 can be labeled by 68Ga for PET imaging. 68Ga-NODAGA-LM3 is a SSTR2 antagonist, and can be used for imaging of SSTR positive paragangliomas.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

NODAGA-LM3 Chemical Structure

NODAGA-LM3 Chemical Structure

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500 μg USD 445 In-stock
1 mg USD 710 In-stock
5 mg USD 1780 In-stock
10 mg USD 2850 In-stock
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Based on 1 publication(s) in Google Scholar

Other Forms of NODAGA-LM3:

NODAGA-LM3 Related Antibodies

Top Publications Citing Use of Products

View All Somatostatin Receptor Isoform Specific Products:

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SSTR1 SSTR2 SSTR3 SSTR5 SSTR4

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Description

NODAGA-LM3 can be labeled by 68Ga for PET imaging. 68Ga-NODAGA-LM3 is a SSTR2 antagonist, and can be used for imaging of SSTR positive paragangliomas[1][2].

IC50 & Target[1]

SSTR2

 

Molecular Weight

1521.11

Formula

C68H90ClN15O19S2
Appearance

Solid

Color

White to off-white

Sequence

{NODAGA}-{p-Cl-Phe}-{d-Cys}-Tyr-{d-Phe(4-amino-carbamoyl)}-Lys-Thr-Cys-{d-Tyr}-NH2 (Disulfide bridge: Cys2-Cys7)
Sequence Shortening

{NODAGA}-{p-Cl-Phe}-{d-Cys}-Y-{d-Phe(4-amino-carbamoyl)}-KTC-{d-Tyr}-NH2 (Disulfide bridge: Cys2-Cys7)
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Sealed storage, away from moisture

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

Solvent & Solubility
In Vitro: 

DMSO : 66.67 mg/mL (43.83 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 0.6574 mL 3.2871 mL 6.5741 mL
5 mM 0.1315 mL 0.6574 mL 1.3148 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
=
Concentration
×
Volume
×
Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

×
Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

Dosage

mg/kg

Animal weight
(per animal)

g

Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 0.6574 mL 3.2871 mL 6.5741 mL 16.4354 mL
5 mM 0.1315 mL 0.6574 mL 1.3148 mL 3.2871 mL
10 mM 0.0657 mL 0.3287 mL 0.6574 mL 1.6435 mL
15 mM 0.0438 mL 0.2191 mL 0.4383 mL 1.0957 mL
20 mM 0.0329 mL 0.1644 mL 0.3287 mL 0.8218 mL
25 mM 0.0263 mL 0.1315 mL 0.2630 mL 0.6574 mL
30 mM 0.0219 mL 0.1096 mL 0.2191 mL 0.5478 mL
40 mM 0.0164 mL 0.0822 mL 0.1644 mL 0.4109 mL
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NODAGA-LM3 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

NODAGA-LM3Somatostatin ReceptorSSTRsSSTRparagangliomasPET68GaInhibitorinhibitorinhibit

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