1. Signaling Pathways
  2. GPCR/G Protein
    Neuronal Signaling
  3. Somatostatin Receptor
  4. Somatostatin Receptor Inhibitors

Somatostatin Receptor Inhibitors

SSTR1

SSTR2

SSTR3

SSTR5

SSTR4

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Somatostatin Receptor Inhibitors, Agonists, Antagonists & Activators
Product Name SSTR1 SSTR2 SSTR3 SSTR5 SSTR4 Purity
Octreotide  
SSTR2
SSTR3
SSTR5
  99.64%
Cortistatin-14
SSTR1
SSTR2
SSTR3
SSTR5
SSTR4
99.92%
CYN 154806 TFA  
SSTR2
      99.81%
Cyclosomatostatin
SSTR1
        99.52%
CYN 154806  
SSTR2
      99.76%
BIM-23056    
SSTR3
SSTR5
  99.94%
BIM-23190 hydrochloride  
SSTR2
 
SSTR5
  99.64%
TT-232
SSTR1
     
SSTR4
98.27%
Somatostatin-28 (sheep, human rat mouse)      
SSTR5
  99.40%
CH 275
SSTR1
        99.71%
PRL 2915
hsst1, Ki: >1000 nM
hsst2, Ki: 12 nM
hsst2, IC50: 1.8 nM (rat antagonist bioassay versus somatostatin)
hsst3, Ki: 100 nM
hsst5, Ki: 520 nM
hsst4, Ki: 895 nM
99.57%
Cortistatin-29 (reduced)
SSTR1, IC50: 2.8 nM
SSTR2, IC50: 7.1 nM
SSTR3, IC50: 0.2 nM
SSTR5, IC50: 13.7 nM
SSTR4, IC50: 3.0 nM
99.22%
Veldoreotide TFA  
SSTR2, EC50: 37.6 nM
SSTR3, EC50: 31.3 nM
 
SSTR4, EC50: 10.5 nM
98.37%
Veldoreotide  
SSTR2, EC50: 37.6 nM
SSTR3, EC50: 31.3 nM
 
SSTR4, EC50: 10.5 nM
NODAGA-LM3 TFA  
SSTR2
     
NODAGA-LM3  
SSTR2
      99.33%
PRL 3195
hsst1, Ki: 1000 nM
hsst2, Ki: 17 nM
hsst3, Ki: 66 nM
hsst5, Ki: 6 nM
hsst4, Ki: 1000 nM
[Tyr1]-Somatostatin-14  
SSTR2
     
BIM-23056 TFA    
SSTR3
SSTR5
 
BIM-23190  
SSTR2
 
SSTR5
 
Octreotide pamoate  
SSTR2
SSTR3
SSTR5
 
sst2 Receptor agonist-1  
SSTR2, Ki: 0.025 nM
SSTR2, IC50: 4.8 nM
     
Seglitide  
SSTR2
     
Satoreotide  
SSTR2
     
Cortistatin-29
SSTR1, IC50: 2.8 nM
SSTR2, IC50: 7.1 nM
SSTR3, IC50: 0.2 nM
SSTR5, IC50: 13.7 nM
SSTR4, IC50: 3.0 nM
Onzigolide  
SSTR2
     
AP102  
SSTR2, IC50: 0.63 nM
 
SSTR5, IC50: 0.65 nM
 
L-796,778    
SSTR3