Somatostatin Receptor Inhibitors

SSTR1

SSTR2

SSTR3

SSTR5

SSTR4

Somatostatin Receptor Inhibitors, Agonists, Antagonists & Activators

Product Name	SSTR1	SSTR2	SSTR3	SSTR5	SSTR4	Purity
Octreotide		SSTR2	SSTR3	SSTR5		99.64%
Veldoreotide TFA		SSTR2, EC₅₀: 37.6 nM	SSTR3, EC₅₀: 31.3 nM		SSTR4, EC₅₀: 10.5 nM	98.37%
CYN 154806 TFA		SSTR2				99.81%
Cyclosomatostatin	SSTR1					99.52%
BIM-23056			SSTR3	SSTR5		99.94%
TT-232	SSTR1				SSTR4	98.96%
PRL 2915	hsst₁, Ki: >1000 nM	hsst₂, Ki: 12 nM hsst₂, IC₅₀: 1.8 nM (rat antagonist bioassay versus somatostatin)	hsst₃, Ki: 100 nM	hsst₅, Ki: 520 nM	hsst₄, Ki: 895 nM	99.57%
CH 275	SSTR1					99.71%
BIM-23190 hydrochloride		SSTR2		SSTR5		99.64%
Cortistatin-29 (reduced)	SSTR1, IC₅₀: 2.8 nM	SSTR2, IC₅₀: 7.1 nM	SSTR3, IC₅₀: 0.2 nM	SSTR5, IC₅₀: 13.7 nM	SSTR4, IC₅₀: 3.0 nM	99.22%
Somatostatin-28 (sheep, human rat mouse)				SSTR5		99.40%
Veldoreotide		SSTR2, EC₅₀: 37.6 nM	SSTR3, EC₅₀: 31.3 nM		SSTR4, EC₅₀: 10.5 nM
NODAGA-LM3 TFA		SSTR2
PRL 3195	hsst₁, Ki: 1000 nM	hsst₂, Ki: 17 nM	hsst₃, Ki: 66 nM	hsst₅, Ki: 6 nM	hsst₄, Ki: 1000 nM
[Tyr1]-Somatostatin-14		SSTR2
BIM-23056 TFA			SSTR3	SSTR5
BIM-23190		SSTR2		SSTR5
Octreotide pamoate		SSTR2	SSTR3	SSTR5
sst2 Receptor agonist-1		SSTR2, Ki: 0.025 nM SSTR2, IC₅₀: 4.8 nM
Seglitide		SSTR2
Satoreotide		SSTR2
NODAGA-LM3		SSTR2
Cortistatin-29	SSTR1, IC₅₀: 2.8 nM	SSTR2, IC₅₀: 7.1 nM	SSTR3, IC₅₀: 0.2 nM	SSTR5, IC₅₀: 13.7 nM	SSTR4, IC₅₀: 3.0 nM
Onzigolide		SSTR2
AP102		SSTR2, IC₅₀: 0.63 nM		SSTR5, IC₅₀: 0.65 nM
L-796,778			SSTR3

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