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beta-adrenoceptor

" in MedChemExpress (MCE) Product Catalog:

By Targets:	5-HT Receptor (14) Adrenergic Receptor (46) Akt (2) Angiotensin Receptor (2) Angiotensin-converting Enzyme (ACE) (1) Bcl-2 Family (1) Calcium Channel (1) Caspase (1) Cholinesterase (ChE) (1) Drug Metabolite (3) Endogenous Metabolite (1) GABA Receptor (1) Isotope-Labeled Compounds (3) mAChR (1) PI3K (2) Renin (3)
By Research Areas:	Cancer (7) Cardiovascular Disease (32) Endocrinology (23) Inflammation/Immunology (3) Metabolic Disease (1) Neurological Disease (18)
Click Chemistry:	Alkynes (1)

Inhibitors & Agonists

Peptides

Natural
Products

Isotope-Labeled Compounds

Click Chemistry

Targets Recommended: Amyloid-β TGF-β Receptor Beta-secretase β-glucuronidase TGF-beta/Smad 17β-HSD β-catenin 11β-HSD Beta-lactamase Dopamine β-hydroxylase

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-100635

Diacetolol	Drug Metabolite	Cardiovascular Disease Endocrinology
Diacetolol is an active metabolite of the beta-adrenoceptor blocking agent Acebutolol (HY-17497) .

HY-17501A

Bambuterol hydrochloride 1 Publications Verification (±)-Bambuterol hydrochloride; KWD-2183 hydrochloride	Adrenergic Receptor	Endocrinology
Bambuterol hydrochloride ((±)-Bambuterol hydrochloride; KWD-2183 hydrochloride) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a proagent of terbutaline.

HY-128379

Labetalone hydrochloride	Drug Metabolite	Others
Labetalone hydrochloride is an impurity of Labetalol. Labetalol is an orally active adrenoceptor blocking agent which is a competitive antagonist at both alpha- and beta-adrenoceptor sites .

HY-17501S

Bambuterol-d9 hydrochloride (±)-Bambuterol-d₉ hydrochloride; KWD-2183-d₉ hydrochloride	Adrenergic Receptor	Endocrinology
Bambuterol-d₉ (hydrochloride) is the deuterium labeled Bambuterol. Bambuterol ((±)-Bambuterol) hydrochloride is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a prodrug of terbutaline.

HY-U00019

Pamatolol	Adrenergic Receptor	Cardiovascular Disease Endocrinology
Pamatolol is a cardioselective *beta-adrenoceptor* antagonist without sympathomimetic activity.

HY-106361

Flerobuterol CRL 40827	Adrenergic Receptor	Neurological Disease
Flerobuterol is a *beta-adrenoceptor* agonist with antidepressant activity. Flerobuterol enhances serotonergic neurotransmission .

HY-106361A

Flerobuterol hydrochloride CRL 40827 hydrochloride	Adrenergic Receptor	Neurological Disease
Flerobuterol hydrochloride is a *beta-adrenoceptor* agonist with antidepressant activity. Flerobuterol hydrochloride enhances serotonergic neurotransmission .

HY-U00356

Tertatolol (±)-Tertatolol; Racemic Tertatolol; dl-Tertatolol	Adrenergic Receptor 5-HT Receptor	Cardiovascular Disease Endocrinology
Tertatolol is a potent antagonist of *beta-adrenoceptor* and 5-HT receptor, with unique renal vasodilatatory effects.

HY-17501

Bambuterol (±)-Bambuterol; KWD-2183	Adrenergic Receptor	Endocrinology
Bambuterol ((±)-Bambuterol; KWD-2183) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a proagent of terbutaline.

HY-19578B

Isamoltane hemifumarate (±)-Isamoltane hemifumarate	5-HT Receptor Adrenergic Receptor	Neurological Disease
Isamoltane hemifumarate is a selective antagonist of 5-HT_1B receptor, with an IC₅₀ of 39 nM for inhibits the binding of [ ¹²⁵I]ICYP to 5-HT_1B recognition sites in rat brain membranes. Isamoltane hemifumarate is also a *β-adrenoceptor* ligand, with an IC₅₀ of 8.4 nM. Isamoltane hemifumarate shows anxiolytic activity .

HY-17501AR

Bambuterol hydrochloride (Standard)	Adrenergic Receptor	Endocrinology
Bambuterol hydrochloride (Standard) is the analytical standard of Bambuterol hydrochloride. This product is intended for research and analytical applications. Bambuterol hydrochloride ((±)-Bambuterol hydrochloride; KWD-2183 hydrochloride) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a proagent of terbutaline.

HY-128379R

Labetalone hydrochloride (Standard)	Drug Metabolite	Others
Labetalone (hydrochloride) (Standard) is the analytical standard of Labetalone (hydrochloride). This product is intended for research and analytical applications. Labetalone hydrochloride is an impurity of Labetalol. Labetalol is an orally active adrenoceptor blocking agent which is a competitive antagonist at both alpha- and beta-adrenoceptor sites .

HY-B0010B

Formoterol-1 (±)Formoterol	Adrenergic Receptor	Inflammation/Immunology
Formoterol ((±)Formoterol) is an orally active β2-selective agonist. Formoterol potently relaxes the peripheral airways through stimulating the beta 2-adrenoceptors selectively as is the case in the central airways and that it significantly inhibits IgE-mediated slow reactive substance of anaphylaxis (SRS-A) release through beta-adrenoceptor stimulation .

HY-101752

(±)-Befunolol	Adrenergic Receptor	Cardiovascular Disease Endocrinology
(±)-Befunolol is a *β-adrenoceptor* blocking agent.

HY-101752A

(±)-Befunolol hydrochloride	Adrenergic Receptor	Cardiovascular Disease Endocrinology
(±)-Befunolol hydrochloride is a *β-adrenoceptor* blocking agent.

HY-19673

KUL-7211	Adrenergic Receptor	Endocrinology
KUL 7211 is a selective *β-adrenoceptor* agonist.

HY-121692A

(S)-Alprenolol L-tartrate	Adrenergic Receptor	Cardiovascular Disease
(S)-Alprenolol is a potent and nonselective *β-adrenoceptor* antagonist .

HY-121843

Ronactolol	Adrenergic Receptor	Endocrinology
Ronactolol, an aminopropanol derivative with β-adrenoceptor blocking activity .

HY-106499

Sulfinalol	Adrenergic Receptor	Cardiovascular Disease
Sulfinalol is an orally active *β-adrenoceptor* antagonist with direct vasodilator activity .

HY-B1670A

(-)-Isoproterenol hydrochloride Levisoprenaline hydrochloride; Proternol L hydrochloride	Adrenergic Receptor	Cardiovascular Disease
(-)-Isoproterenol (Levisoprenaline; Proternol L) hydrochloride is a *β-adrenoceptor* agonist. (-)-Isoproterenol induces ventricular remodeling .

HY-106499A

Sulfinalol hydrochloride	Adrenergic Receptor	Cardiovascular Disease
Sulfinalol hydrochloride is an orally active *β-adrenoceptor* antagonist with direct vasodilator activity. Sulfinalol hydrochloride is an antihypertensive agent .

HY-19673A

KUL-7211 racemate	Adrenergic Receptor	Endocrinology
KUL-7211 racemate is the racemate of KUL-7211. KUL-7211 is a selective *β-adrenoceptor* agonist .

HY-A0252

Bupranolol	Adrenergic Receptor	Inflammation/Immunology Cancer
Bupranolol is an orally active, competitive and non-selective *β-adrenoceptor* antagonist without intrinsic sympathomimetic activity .

HY-W181626

Tiprenolol DU 21445	5-HT Receptor	Cardiovascular Disease
Tiprenolol is a *β-adrenoceptor* blocker. Tiprenolol can abolish the ventricular arrhythmias produced by adrenaline in dogs respired with halothane .

HY-W181626A

Tiprenolol hydrochloride DU 21445 hydrochloride	5-HT Receptor	Cardiovascular Disease
Tiprenolol hydrochloride is a β-adrenoceptor blocker. Tiprenolol hydrochloride abolished ventricular arrhythmias induced by intravenous epinephrine in dogs receiving halothane inhalation .

HY-116790A

(+)-Penbutolol (R)-Penbutolol; (+)-Isopenbutolol	Adrenergic Receptor	Metabolic Disease Endocrinology
(+)-Penbutolol is a β-adrenoceptor antagonist, with an IC₅₀ of 0.74 μM . (+)-Penbutolol is an optical isomer of l-penbutolol with Na ⁺ channel-blocking action .

HY-120939

S14063	5-HT Receptor	Neurological Disease
S14063 is a potent 5-HT1A receptor antagonist. S14063 is devoid of β-adrenoceptor blocking properties .

HY-100635S

Diacetolol-d7	Isotope-Labeled Compounds Adrenergic Receptor	Cardiovascular Disease Endocrinology
Diacetolol-d₇ is a deuterium labeled Diacetolol. Diacetolol is the major metabolite of Acebutolol. Diacetolol is a β-adrenoceptor blocking and anti-arrhythmic agent[1].

HY-108302

Nifenalol	Adrenergic Receptor	Others
Nifenalol is a β-adrenergic receptor blocker. Nifenalol inhibits β-adrenoceptor differentiation in right atrium, diaphragm and adipose tissue in a rat model .

HY-17495

Carteolol OPC-1085	Adrenergic Receptor Caspase Bcl-2 Family	Neurological Disease
Carteolol is a non-selective *β-adrenoceptor* antagonist. Carteolol induces apoptosis via a caspase activated and mitochondrial-dependent pathway. Carteolol can be used for glaucoma research .

HY-U00183

Epanolol Visacor; ICI141292	Adrenergic Receptor	Cardiovascular Disease Endocrinology
Epanolol (Visacor; ICI141292) is a potent *β-adrenoceptor* partial agonist with a greater affinity for β1- than β2-adrenoceptors.

HY-103207

Amibegron hydrochloride SR 58611A	Adrenergic Receptor	Neurological Disease Endocrinology
Amibegron hydrochloride is a selective *β3-adrenoceptor* agonist, with an EC₅₀ of 3.5 nM for *β-adrenoceptor* in rat colon; Amibegron hydrochloride has anxiolytic and antidepressant activity.

HY-111479

Amibegron SR-58611	Adrenergic Receptor	Neurological Disease Endocrinology
Amibegron is a selective *β3-adrenoceptor* agonist, with an EC₅₀ of 3.5 nM for *β-adrenoceptor* in rat colon; Amibegron has anxiolytic and antidepressant activity.

HY-A0252R

Bupranolol (Standard)	Adrenergic Receptor	Inflammation/Immunology Cancer
Bupranolol (Standard) is the analytical standard of Bupranolol. This product is intended for research and analytical applications. Bupranolol is an orally active, competitive and non-selective *β-adrenoceptor* antagonist without intrinsic sympathomimetic activity .

HY-101721

Ko-3290	Adrenergic Receptor	Cardiovascular Disease Endocrinology
Ko-3290 is an antagonist of *β-adrenoceptor*, with cardioselectivity and antilipolytic effects in animals. Ko-3290 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

HY-P1376

G-Protein antagonist peptide	mAChR Adrenergic Receptor	Endocrinology
G-Protein antagonist peptide is the substance P-related peptide that inhibits binding of G proteins to their receptors. G-Protein antagonist peptide competitively and reversibly inhibits M2 muscarinic receptor activation of G_i or G_o and inhibits G_s activation by β-adrenoceptors.

HY-100606

l-Pindolol (-)-Pindolol; (S)-(-)-Pindolol; S-Pindolol	5-HT Receptor Adrenergic Receptor	Neurological Disease
l-Pindolol ((-)-pindolol) is a reversible, competitive and orally active 5-HT1A/1B antagonist. l-Pindolol is a partial *β-adrenoceptor* agonist. l-Pindolol can be used for the research of neurological disease .

HY-17380

(S)-Timolol maleate 2 Publications Verification (S)-L-714,465 maleate; MK 950	Adrenergic Receptor	Cardiovascular Disease Neurological Disease Cancer
(S)-Timolol Maleate (L-714,465 Maleate) is a non-cardioselective hydrophilic *β-adrenoceptor* blocker. (S)-Timolol Maleate is widely used as standard medication for intraocular pressure (glaucoma) by preventing the production of aqueous humor. (S)-Timolol Maleate can be used for hypertension, angina pectoris and myocardial infarction .

HY-B1517B

Alprenolol benzoate	5-HT Receptor	Cardiovascular Disease Cancer
Alprenolol benzoate is an orally active non-selective *β-adrenoceptor* antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol benzoate is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent .

HY-A0295

(R)-Propranolol hydrochloride	Adrenergic Receptor	Cardiovascular Disease Neurological Disease Endocrinology
(R)-Propranolol hydrochloride is a less active enantiomer of the β-adrenoceptor antagonist propranolol (HY-B0573). Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β₁AR and β₂AR with K_i values of 1.8 nM and 0.8 nM, respectively .

HY-116790

(-)-Penbutolol (S)-Penbutolol; (-)-Isopenbutolol	Adrenergic Receptor 5-HT Receptor	Neurological Disease Endocrinology
(-)-Penbutolol ((S)-Penbutolol) is a potent *β-adrenoceptor* and 5-HT receptor antagonist with K_i values of 11.6 nM and 11.9 nM for 5-HT in rat cornu ammonis 1 (CA1) and human CA3. (-)-Penbutolol can increase hippocampal 5-HT output .

HY-B1517

Alprenolol 5+ Cited Publications (RS)-Alprenolol; dl-Alprenolol	5-HT Receptor	Cardiovascular Disease Cancer
Alprenolol ((RS)-Alprenolol; dl-Alprenolol) is an orally active non-selective *β-adrenoceptor* antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent .

HY-B1517A

Alprenolol hydrochloride 5+ Cited Publications (RS)-Alprenolol hydrochloride; dl-Alprenolol hydrochloride	5-HT Receptor	Cardiovascular Disease Cancer
Alprenolol ((RS)-Alprenolol; dl-Alprenolol) hydrochloride is an orally active non-selective *β-adrenoceptor* antagonist and an antagonist of 5-HT1A and 5-HT1B receptors. Alprenolol hydrochloride is used as an anti-hypertensive, anti-anginal and anti-arrhythmic agent .

HY-111013

VK-II-86	Others	Cardiovascular Disease
VK-II-86 is a Carvedilol (HY-B0006) analogue lacking antagonist activity at β-adrenoceptors, in hypokalaemia. VK-II-86 prevents hypokalaemia-induced ventricular arrhythmia through multi-channel effects. VK-II-86 prevents all hypokalaemia-induced changes in ion channel activity and oxidative stress .

HY-16056

Arbutamine	Adrenergic Receptor	Cardiovascular Disease
Arbutamine is a short-acting, potent and nonselective *β-adrenoceptor* agonist. Arbutamine stimulates cardiac β₁-, tracheal β₂-, and adiopocyte β₃- adrenergic receptors. Arbutamine provides cardiac stress increases heart rate, cardiac contractility, and systolic blood pressure. Arbutamine can be used for cardiac stress agent .

HY-16056A

Arbutamine hydrochloride	Adrenergic Receptor	Cardiovascular Disease
Arbutamine hydrochloride is a short-acting, potent and nonselective *β-adrenoceptor* agonist. Arbutamine hydrochloride stimulates cardiac β₁-, tracheal β₂-, and adiopocyte β₃- adrenergic receptors. Arbutamine hydrochloride provides cardiac stress increases heart rate, cardiac contractility, and systolic blood pressure. Arbutamine hydrochloride can be used for cardiac stress agent .

HY-P5189A

*His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA*	Endogenous Metabolite Cholinesterase (ChE)	Others
His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA, is a growth hormone releasing peptide, as well as a metabolite of GHRP-1. GHRP-1, or Ala-His-D-beta Nal-Ala-Trp-D-Phe-Lys-NH2, has the effect of promoting the release of growth hormone (GH). GHRP-1 increases GH release and increases [Ca2+]i levels in static monolayer cells of rat pituitary gland, but does not affect cAMP levels .

HY-17494S

(Rac)-Timolol-d5 maleate (Rac)-L-714,465-d₅ maleate; (Rac)-MK 950-d₅	Isotope-Labeled Compounds Adrenergic Receptor	Cardiovascular Disease Neurological Disease
rac Timolol-d₅ (maleate) is a labelled racemic (S)-Timolol maleate. (S)-Timolol Maleate (L-714,465 Maleate) is a non-cardioselective hydrophilic β-adrenoceptor blocker. (S)-Timolol Maleate is widely used as standard medication for intraocular pressure (glaucoma) by preventing the production of aqueous humor. (S)-Timolol Maleate can be used for hypertension, angina pectoris and myocardial infarction[1][2][3].

HY-17380S

(S)-Timolol-d9 maleate (S)-L-714,465-d₉ maleate; MK 950-d₉	Isotope-Labeled Compounds Adrenergic Receptor	Cardiovascular Disease Neurological Disease
(S)-Timolol-d₉ (maleate) is deuterium labeled (S)-Timolol (Maleate). (S)-Timolol Maleate (L-714,465 Maleate) is a non-cardioselective hydrophilic β-adrenoceptor blocker. (S)-Timolol Maleate is widely used as standard medication for intraocular pressure (glaucoma) by preventing the production of aqueous humor. (S)-Timolol Maleate can be used for hypertension, angina pectoris and myocardial infarction[1][2][3].

HY-17380R

(S)-Timolol maleate (Standard) (S)-L-714,465 maleate (Standard); MK 950 (Standard)	Adrenergic Receptor	Cardiovascular Disease Neurological Disease
(S)-Timolol (maleate) (Standard) is the analytical standard of (S)-Timolol (maleate). This product is intended for research and analytical applications. (S)-Timolol Maleate (L-714,465 Maleate) is a non-cardioselective hydrophilic *β-adrenoceptor* blocker. (S)-Timolol Maleate is widely used as standard medication for intraocular pressure (glaucoma) by preventing the production of aqueous humor. (S)-Timolol Maleate can be used for hypertension, angina pectoris and myocardial infarction .

Cat. No.	Product Name	Target	Research Area

HY-P4285

β-Aspartylalanine	Peptides	Others
β-Aspartylalanine is a substrate for β-aspartyl peptidase and used to measure β-aspartyl peptidase activity in fecal supernatants .

HY-P1376

G-Protein antagonist peptide	mAChR Adrenergic Receptor	Endocrinology
G-Protein antagonist peptide is the substance P-related peptide that inhibits binding of G proteins to their receptors. G-Protein antagonist peptide competitively and reversibly inhibits M2 muscarinic receptor activation of G_i or G_o and inhibits G_s activation by β-adrenoceptors.

HY-P5189A

*His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA*	Endogenous Metabolite Cholinesterase (ChE)	Others
His-D-beta-Nal-Ala-Trp-D-Phe-Lys-NH2 TFA, is a growth hormone releasing peptide, as well as a metabolite of GHRP-1. GHRP-1, or Ala-His-D-beta Nal-Ala-Trp-D-Phe-Lys-NH2, has the effect of promoting the release of growth hormone (GH). GHRP-1 increases GH release and increases [Ca2+]i levels in static monolayer cells of rat pituitary gland, but does not affect cAMP levels .

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-17501

Bambuterol (±)-Bambuterol; KWD-2183	Classification of Application Fields Disease Research Fields Endocrinology	Adrenergic Receptor
Bambuterol ((±)-Bambuterol; KWD-2183) is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a proagent of terbutaline.

Cat. No.	Product Name	Chemical Structure

HY-17501S

Bambuterol-d9 hydrochloride
Bambuterol-d₉ (hydrochloride) is the deuterium labeled Bambuterol. Bambuterol ((±)-Bambuterol) hydrochloride is a long acting beta-adrenoceptor agonist (LABA) used in the treatment of asthma; it also is a prodrug of terbutaline.

HY-17494S

(Rac)-Timolol-d5 maleate

rac Timolol-d₅ (maleate) is a labelled racemic (S)-Timolol maleate. (S)-Timolol Maleate (L-714,465 Maleate) is a non-cardioselective hydrophilic β-adrenoceptor blocker. (S)-Timolol Maleate is widely used as standard medication for intraocular pressure (glaucoma) by preventing the production of aqueous humor. (S)-Timolol Maleate can be used for hypertension, angina pectoris and myocardial infarction[1][2][3].

HY-100635S

Diacetolol-d7
Diacetolol-d₇ is a deuterium labeled Diacetolol. Diacetolol is the major metabolite of Acebutolol. Diacetolol is a β-adrenoceptor blocking and anti-arrhythmic agent[1].

HY-17380S

(S)-Timolol-d9 maleate

(S)-Timolol-d₉ (maleate) is deuterium labeled (S)-Timolol (Maleate). (S)-Timolol Maleate (L-714,465 Maleate) is a non-cardioselective hydrophilic β-adrenoceptor blocker. (S)-Timolol Maleate is widely used as standard medication for intraocular pressure (glaucoma) by preventing the production of aqueous humor. (S)-Timolol Maleate can be used for hypertension, angina pectoris and myocardial infarction[1][2][3].

Cat. No.	Product Name		Classification

HY-101721

Ko-3290		Alkynes
Ko-3290 is an antagonist of *β-adrenoceptor*, with cardioselectivity and antilipolytic effects in animals. Ko-3290 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

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