1. Signaling Pathways
  2. Vitamin D Related/Nuclear Receptor
  3. Nuclear Hormone Receptor 4A/NR4A
  4. Nuclear Hormone Receptor 4A/NR4A Inhibitors

Nuclear Hormone Receptor 4A/NR4A Inhibitors

Nur77/NR4A1

Nurr1/NR4A2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Nuclear Hormone Receptor 4A/NR4A Inducers, Agonists, Antagonists & Activators
Product Name Nur77/NR4A1 Nurr1/NR4A2 Purity
Cytosporone B
Nur77/NR4A1
  98.63%
DIM-C-pPhOH
Nur77/NR4A1
  99.05%
Teduglutide
Nur77/NR4A1
  99.94%
Amodiaquine  
Nurr1/NR4A2
99.98%
Amodiaquine dihydrochloride dihydrate  
Nurr1/NR4A2
99.89%
Nurr1 agonist 12  
Nurr1/NR4A2, EC50: 0.06 μM
Amodiaquine dihydrochloride  
Nurr1/NR4A2
99.89%
DIM-C-pPhCO2Me
Nur77/NR4A1
  99.47%
TMPA
Nur77/NR4A1
  98.22%
C-DIM12  
Nurr1/NR4A2
98.32%
Nurr1 agonist 2  
Nurr1/NR4A2
99.27%
Triptohypol C
Nur77/NR4A1
 
4A7C-301  
Nurr1/NR4A2
99.86%
DIM-C-pPhOCH3
Nur77/NR4A1
  99.49%
4-PQBH
Nur77/NR4A1
  99.08%
IP7e  
Nurr1/NR4A2
99.65%
Nurr1 inverse agonist-1  
Nurr1/NR4A2
99.79%
THPN
Nur77/NR4A1
  98.00%
Nur77 modulator 1
Nur77/NR4A1
  98.61%
Nur77 modulator 4
Nur77/NR4A1, Kd: 0.477 μM
 
Nur77 modulator 2
Nur77/NR4A1
 
Nur77 antagonist 1
Nur77/NR4A1
 
Nurr1 agonist 9  
Nurr1/NR4A2, EC50: 0.09 μM
Nurr1/NR4A2, Ki: 0.17 μM
Nurr1 agonist 10  
Nurr1/NR4A2, EC50: 40 nM
Nurr1 agonist 5  
Nurr1/NR4A2