2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor 5-HT Receptor
  4. Cyanopindolol

Cyanopindolol is an β3-adrenoceptor antagonist. Cyanopindolol is a potent and selective antagonist at the presynaptic serotonin autoreceptor in the rat brain cortex. Cyanopindolol has binding affinity for 5-HT1A and 5-HT1B receptor (Ki: 2.1 and 3 nM respectively).

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Cyanopindolol Chemical Structure

Cyanopindolol Chemical Structure

CAS No. : 69906-85-0

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Other Forms of Cyanopindolol:

Cyanopindolol Related Antibodies

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Description

Cyanopindolol is an β3-adrenoceptor antagonist. Cyanopindolol is a potent and selective antagonist at the presynaptic serotonin autoreceptor in the rat brain cortex. Cyanopindolol has binding affinity for 5-HT1A and 5-HT1B receptor (Ki: 2.1 and 3 nM respectively)[1][2][3].

IC50 & Target[3]

β3 adrenoceptor

 

5-HT1A Receptor

2.1 nM (Ki)

5-HT1B Receptor

3 nM (Ki)

Molecular Weight

287.36

Formula

C16H21N3O2
CAS No.
SMILES

CC(C)(NCC(O)COC1=CC=CC2=C1C=C(C#N)N2)C
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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Cyanopindolol Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Cyanopindolol69906-85-0Adrenergic Receptor5-HT ReceptorBeta ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorserotoninAdrenergic receptorInhibitorinhibitorinhibit

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