2. Metabolic Enzyme/Protease Vitamin D Related/Nuclear Receptor
  3. RAR/RXR
  4. RARα antagonist 1

RARα antagonist 1 (compound 21) is an orally active and selective retinoic acid receptor α(RARα) antagonist, with the IC50 of 4.6nM.

For research use only. We do not sell to patients.

RARα antagonist 1 Chemical Structure

RARα antagonist 1 Chemical Structure

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RARα antagonist 1 Related Antibodies

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Description

RARα antagonist 1 (compound 21) is an orally active and selective retinoic acid receptor α(RARα) antagonist, with the IC50 of 4.6nM[1].

IC50 & Target

4.6nM (RARα)[1]
Molecular Weight

413.47

Formula

C26H23NO4
SMILES

OC(C1=CC=C(NC(C(C=C2)=CC3=C2OC(C)(C)C=C3C4=CC=C(C)C=C4)=O)C=C1)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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RARα antagonist 1 Related Classifications

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

RARα antagonist 1RARα antagonist1RARα antagonist-1RAR/RXRRetinoic acid receptorsRetinoid X receptorsretinoic acid receptor αorally activeRara?/? male micemetabolic stabilityInhibitorinhibitorinhibit

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RARα antagonist 1
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