2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. SB251023

SB251023 is a β3-adrenergic receptor agonist with pEC50 values of 7.14 and 6.91 for the β3a- and β3b-adrenergic receptors, respectively. SB251023 is capable of modulating cyclic AMP levels and extracellular acidification rate (EAR) in cells. It has potential application value in the study of cardiovascular diseases and metabolic-related disorders.

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SB251023 Chemical Structure

SB251023 Chemical Structure

CAS No. : 208842-53-9

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SB251023 Related Antibodies

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Description

SB251023 is a β3-adrenergic receptor agonist with pEC50 values of 7.14 and 6.91 for the β3a- and β3b-adrenergic receptors, respectively. SB251023 is capable of modulating cyclic AMP levels and extracellular acidification rate (EAR) in cells. It has potential application value in the study of cardiovascular diseases and metabolic-related disorders[1].

IC50 & Target

Beta-3 adrenergic receptor

 

Molecular Weight

511.55

Formula

C28H34NO6P
CAS No.
SMILES

O=P(COC1=CC=C(C=C1)CC2(CCCC2)NC[C@@H](COC3=CC=C(C=C3)O)O)(O)C4=CC=CC=C4
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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SB251023 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

SB251023208842-53-9SB 251023SB-251023Adrenergic ReceptorBeta ReceptorInhibitorinhibitorinhibit

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